FAIRMol

OSA_Lib_90

Pose ID 35953 Compound 2831 Pose 1312

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.742 kcal/mol/HA) ✓ Good fit quality (FQ -6.83) ✓ Good H-bonds (3 bonds) ✗ High strain energy (15.6 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-19.280
kcal/mol
LE
-0.742
kcal/mol/HA
Fit Quality
-6.83
FQ (Leeson)
HAC
26
heavy atoms
MW
349
Da
LogP
2.40
cLogP
Strain ΔE
15.6 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 21 π–π 0 Clashes 2 Severe clashes 0
Final rank3.04881531146618Score-19.2797
Inter norm-0.789224Intra norm0.047696
Top1000noExcludedno
Contacts13H-bonds3
Artifact reasongeometry warning; 12 clashes; 2 protein contact clashes; moderate strain Δ 16.8
ResiduesA:ALA209;A:ALA90;A:ASN208;A:GLY214;A:GLY215;A:LEU73;A:LYS211;A:LYS89;A:MET70;A:PRO212;A:PRO213;A:TYR210;A:VAL88

Protein summary

493 residues
Protein targetT16Atoms7551
Residues493Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:276; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6RB5Contacts12
PoseOpen native poseH-bonds0
IFP residuesA:ALA90; A:ARG74; A:GLY85; A:LEU73; A:LYS89; A:MET70; A:PHE83; A:PRO212; A:PRO213; A:SER86; A:SER87; A:VAL88
Current overlap7Native recall0.58
Jaccard0.39RMSD-
H-bond strict0Strict recall-
H-bond same residue+role0Role recall-
H-bond same residue0Residue recall-

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1312 3.04881531146618 -0.789224 -19.2797 3 13 7 0.58 - - no Current
1324 3.335456433991353 -0.881207 -21.8722 4 13 7 0.58 - - no Open
1315 3.832949461622242 -0.869764 -22.5535 3 14 9 0.75 - - no Open
1322 3.838562660346953 -0.825348 -21.2745 4 12 7 0.58 - - no Open
1318 3.964568238201872 -0.700693 -18.0911 4 10 5 0.42 - - no Open
1326 4.017280272361394 -0.760736 -18.8783 3 13 8 0.67 - - no Open
1313 53.73537365533876 -0.780042 -18.9905 3 13 7 0.58 - - no Open
1320 53.92370550138362 -0.954734 -23.2526 4 13 7 0.58 - - no Open
1321 54.095948950114774 -0.770125 -18.4558 2 13 7 0.58 - - no Open
1323 54.229993089198935 -0.738022 -17.9146 3 12 8 0.67 - - no Open
1316 54.24618337723126 -0.791883 -19.2566 2 14 8 0.67 - - no Open
1325 55.003938327992266 -0.77134 -19.0864 2 13 7 0.58 - - no Open
1327 55.06958616550822 -0.752956 -19.0502 2 15 10 0.83 - - no Open
1314 54.23087636810456 -0.874766 -22.0134 4 12 7 0.58 - - yes Open
1317 55.793383662147505 -0.757032 -16.132 2 14 9 0.75 - - yes Open
1319 57.66482927389143 -0.902158 -21.5772 3 14 8 0.67 - - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -19.280kcal/mol
Ligand efficiency (LE) -0.7415kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.832
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 348.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.40
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 15.56kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 109.93kcal/mol
Minimised FF energy 94.38kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.