FAIRMol

OHD_TB2020_5

Pose ID 3559 Compound 197 Pose 241

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.685 kcal/mol/HA) ✓ Good fit quality (FQ -7.32) ✗ Very high strain energy (47.2 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-30.130
kcal/mol
LE
-0.685
kcal/mol/HA
Fit Quality
-7.32
FQ (Leeson)
HAC
44
heavy atoms
MW
606
Da
LogP
5.37
cLogP
Strain ΔE
47.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: mixed
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 47.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 19 Severe clashes 0
Final rank10.053624366210254Score-30.1296
Inter norm-0.560046Intra norm-0.124716
Top1000noExcludedno
Contacts13H-bonds1
Artifact reasongeometry warning; 14 clashes; 19 protein contact clashes; high strain Δ 45.9
ResiduesA:ARG97;A:ASN58;A:ASP52;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:PHE56;A:PHE91;A:PRO50;A:PRO88;A:THR54;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap10Native recall0.50
Jaccard0.43RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
219 4.6302099942158925 -0.503435 -20.6429 0 19 0 0.00 0.00 - no Open
139 5.794697303459581 -0.392755 -18.0678 3 15 1 0.05 0.00 - no Open
217 6.116056632700398 -0.50366 -23.1694 0 20 0 0.00 0.00 - no Open
247 7.619680315638954 -0.494608 -15.7059 0 17 14 0.70 0.00 - no Open
213 8.172789639007322 -0.580209 -26.3337 3 20 0 0.00 0.00 - no Open
215 9.068038958891496 -0.603154 -21.3249 3 18 0 0.00 0.00 - no Open
140 9.672599851697436 -0.400196 -15.5328 5 18 1 0.05 0.00 - no Open
241 10.053624366210254 -0.560046 -30.1296 1 13 10 0.50 0.00 - no Current
240 7.341478671968607 -0.584644 -25.7145 1 18 16 0.80 0.00 - yes Open
222 8.07721139061682 -0.516534 -17.9777 1 16 0 0.00 0.00 - yes Open
137 8.575914499429317 -0.396661 -16.5688 2 16 1 0.05 0.00 - yes Open
245 8.881429646481902 -0.573363 -19.1523 1 18 16 0.80 0.00 - yes Open
220 9.438224068420311 -0.602712 -19.2251 2 21 0 0.00 0.00 - yes Open
214 9.96079017008822 -0.520144 -26.0539 2 20 0 0.00 0.00 - yes Open
246 10.489749462601512 -0.608072 -18.308 2 20 18 0.90 0.00 - yes Open
216 11.234574649205847 -0.49917 -18.3088 2 20 0 0.00 0.00 - yes Open
244 11.559469917061858 -0.579467 -23.8198 3 14 12 0.60 0.20 - yes Open
242 12.209807756178435 -0.581409 -25.4869 1 21 17 0.85 0.00 - yes Open
221 12.806466053653423 -0.59562 -21.5257 3 18 0 0.00 0.00 - yes Open
218 58.63076534262176 -0.579693 -21.4408 3 16 0 0.00 0.00 - yes Open
138 58.913850953012265 -0.516596 -20.5496 3 15 0 0.00 0.00 - yes Open
243 63.24444273701941 -0.606511 -27.6238 3 15 12 0.60 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -30.130kcal/mol
Ligand efficiency (LE) -0.6848kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.317
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 44HA

Physicochemical properties

Molecular weight 605.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.37
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 47.22kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 177.73kcal/mol
Minimised FF energy 130.51kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.