FAIRMol

OHD_Leishmania_45

Pose ID 3347 Compound 753 Pose 29

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good H-bonds (3 bonds) ✗ Very high strain energy (71.2 kcal/mol) ✗ Poor LE (0.125 kcal/mol/HA) ✗ Poor fit quality (FQ 1.42) ✗ Geometry warnings ℹ SASA not computed
Score
7.260
kcal/mol
LE
0.125
kcal/mol/HA
Fit Quality
1.42
FQ (Leeson)
HAC
58
heavy atoms
MW
811
Da
LogP
0.36
cLogP
Strain ΔE
71.2 kcal/mol
SASA buried
computing…
Overall: Likely artefact or unreliable pose
Binding evidence: weak
Native-like contacts: strong
Ligand efficiency: weak
Geometry reliability: low
Reason: geometry warning, clashes, strain 71.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 1 Clashes 11 Severe clashes 1 ⚠ Hydrophobic exposure 39%
⚠️Partial hydrophobic solvent exposure
39% of hydrophobic surface appears solvent-exposed (16/41 atoms). Partial exposure is common but may limit selectivity and membrane permeability.
Non-polar atoms 41 Buried (contacted) 25 Exposed 16 LogP 0.36 H-bonds 3
Exposed fragments: phenyl (6/6 atoms exposed)phenyl (5/6 atoms exposed)aliphatic chain/group (5 atoms exposed)
Final rank60.31577280944552Score7.25978
Inter norm-0.299852Intra norm0.425021
Top1000noExcludedyes
Contacts20H-bonds3
Artifact reasonexcluded; geometry warning; 27 clashes; 1 protein clash; high raw intra
ResiduesA:ALA32;A:ILE45;A:LEU94;A:LYS57;A:LYS90;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO50;A:PRO88;A:SER44;A:SER86;A:THR54;A:THR83;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap17Native recall0.85
Jaccard0.74RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
9 13.325459258586285 -0.334152 -0.965184 3 18 16 0.80 0.20 - no Open
22 11.760943129336825 -0.299245 -17.339 2 17 14 0.70 0.20 - yes Open
17 12.761484724464736 -0.316773 -1.59097 3 18 14 0.70 0.40 - yes Open
23 59.98052726506786 -0.421552 -17.6506 5 19 12 0.60 0.00 - yes Open
29 60.31577280944552 -0.299852 7.25978 3 20 17 0.85 0.00 - yes Current
26 60.59663818971363 -0.360703 -12.2414 6 17 12 0.60 0.20 - yes Open
12 61.38609649517504 -0.371002 -20.1264 7 15 11 0.55 0.20 - yes Open
13 61.414446497231125 -0.426789 -10.6427 7 15 11 0.55 0.20 - yes Open
11 61.5324330228811 -0.278412 -11.1343 5 14 10 0.50 0.20 - yes Open
16 61.78925105950437 -0.317504 -3.7643 6 20 16 0.80 0.20 - yes Open
8 61.96984000917183 -0.32562 -14.188 4 17 12 0.60 0.00 - yes Open
10 62.14688715416227 -0.392714 -9.15959 3 20 18 0.90 0.20 - yes Open
14 62.35515867735744 -0.450017 -11.4909 4 21 18 0.90 0.00 - yes Open
6 62.879331909694066 -0.461952 -23.5639 7 19 16 0.80 0.20 - yes Open
28 62.88274725756217 -0.46073 -19.3201 5 23 18 0.90 0.20 - yes Open
25 63.27097061699387 -0.292962 -24.042 4 20 17 0.85 0.00 - yes Open
15 64.47132710717256 -0.447251 -8.82597 5 22 14 0.70 0.20 - yes Open
4 64.71227221490146 -0.369835 0.395208 7 16 10 0.50 0.20 - yes Open
18 64.79573960870546 -0.42929 -26.9465 9 21 19 0.95 0.20 - yes Open
31 65.19941468193234 -0.35032 -3.63977 8 16 11 0.55 0.20 - yes Open
30 65.26401004694516 -0.399606 -5.96414 6 18 15 0.75 0.20 - yes Open
3 65.50198510870831 -0.404121 2.84679 8 21 17 0.85 0.20 - yes Open
24 65.62007994550007 -0.36325 -1.63916 5 18 16 0.80 0.00 - yes Open
20 65.80881951412888 -0.313655 -0.785003 3 22 18 0.90 0.00 - yes Open
32 65.96630355466264 -0.394604 0.962119 4 19 17 0.85 0.20 - yes Open
27 66.40733352043566 -0.403614 -6.59538 5 21 18 0.90 0.00 - yes Open
33 66.76375879464149 -0.416966 -9.15118 4 18 16 0.80 0.20 - yes Open
5 67.4612805516657 -0.498199 -10.9711 10 21 18 0.90 0.20 - yes Open
34 68.79246416550914 -0.509692 -11.9263 7 22 18 0.90 0.20 - yes Open
7 69.33706874767066 -0.368499 -1.26329 4 24 19 0.95 0.00 - yes Open
21 70.02141138885924 -0.352638 -13.6495 6 20 16 0.80 0.00 - yes Open
19 75.49517389022188 -0.349628 0.291842 8 25 17 0.85 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score 7.260kcal/mol
Ligand efficiency (LE) 0.1252kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) 1.416
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 58HA

Physicochemical properties

Molecular weight 810.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.36
Lipinski: ≤ 5
Rotatable bonds 13

Conformational strain (MMFF94s)

Strain energy (ΔE) 71.19kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 172.03kcal/mol
Minimised FF energy 100.84kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.