FAIRMol

Z56964630

Pose ID 3265 Compound 140 Pose 3265

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.720 kcal/mol/HA) ✓ Good fit quality (FQ -6.64) ✗ High strain energy (17.2 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-18.729
kcal/mol
LE
-0.720
kcal/mol/HA
Fit Quality
-6.64
FQ (Leeson)
HAC
26
heavy atoms
MW
362
Da
LogP
4.69
cLogP
Strain ΔE
17.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 17.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 5 Severe clashes 1
Final rank4.688739833711961Score-18.7293
Inter norm-0.809414Intra norm0.0890559
Top1000noExcludedyes
Contacts17H-bonds1
Artifact reasonexcluded; geometry warning; 11 clashes; 1 protein clash; moderate strain Δ 13.8
ResiduesA:ALA10;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR137;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap14Native recall0.67
Jaccard0.58RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2556 2.56005718758619 -0.892981 -25.0544 1 19 0 0.00 0.00 - no Open
2299 2.631614367521299 -1.06346 -29.3292 2 15 0 0.00 0.00 - no Open
2554 2.7078098932547885 -0.85633 -21.7921 1 19 0 0.00 0.00 - no Open
2392 3.4007757905046723 -0.89664 -22.5064 3 15 0 0.00 0.00 - no Open
2860 3.459434025282788 -0.586227 -17.2719 1 12 0 0.00 0.00 - no Open
2297 3.864243300287797 -1.0745 -27.8525 2 10 0 0.00 0.00 - no Open
3260 4.208806845415883 -1.06066 -27.9908 1 18 18 0.86 0.20 - no Open
3264 4.23041207454424 -1.0365 -26.874 1 18 18 0.86 0.20 - no Open
2301 4.653312728446953 -1.11181 -27.0313 4 12 0 0.00 0.00 - no Open
2555 5.202364879127718 -0.730112 -18.8269 1 16 0 0.00 0.00 - no Open
2861 5.22955659252202 -0.690301 -13.1113 3 10 0 0.00 0.00 - no Open
2394 5.375966602034466 -0.789683 -21.5239 5 13 0 0.00 0.00 - no Open
2858 5.610705689186814 -0.661211 -16.1929 4 8 0 0.00 0.00 - no Open
2557 6.002580860391582 -0.878923 -18.3346 4 13 0 0.00 0.00 - no Open
3265 4.688739833711961 -0.809414 -18.7293 1 17 14 0.67 0.00 - yes Current
3262 4.8431868433061736 -0.946792 -24.4373 2 17 17 0.81 0.20 - yes Open
2859 5.814987639708491 -0.668481 -16.7205 2 10 0 0.00 0.00 - yes Open
2395 5.956897104524552 -0.856747 -16.9129 5 12 0 0.00 0.00 - yes Open
2393 5.972392960267089 -0.988006 -21.2129 2 16 0 0.00 0.00 - yes Open
3263 8.058799273594556 -0.797034 -18.7622 1 19 18 0.86 0.20 - yes Open
3261 9.365242317841728 -0.879831 -23.8497 1 17 17 0.81 0.00 - yes Open
2302 10.056273785360728 -1.34771 -27.9477 4 18 0 0.00 0.00 - yes Open
2298 10.706812236978191 -1.34102 -29.1209 4 17 0 0.00 0.00 - yes Open
2300 14.113166681221848 -1.25256 -26.7006 2 17 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -18.729kcal/mol
Ligand efficiency (LE) -0.7204kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.637
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 361.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.69
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 17.20kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 72.82kcal/mol
Minimised FF energy 55.62kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.