FAIRMol

Z56175938

Pose ID 3250 Compound 311 Pose 3250

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.867 kcal/mol/HA) ✓ Good fit quality (FQ -7.99) ✗ High strain energy (17.9 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-22.533
kcal/mol
LE
-0.867
kcal/mol/HA
Fit Quality
-7.99
FQ (Leeson)
HAC
26
heavy atoms
MW
362
Da
LogP
5.19
cLogP
Strain ΔE
17.9 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 17.9 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 3 Clashes 12 Severe clashes 2
Final rank8.727101054323805Score-22.5331
Inter norm-0.933372Intra norm0.0667153
Top1000noExcludedyes
Contacts16H-bonds2
Artifact reasonexcluded; geometry warning; 13 clashes; 2 protein clashes; high strain Δ 26.8
ResiduesA:ALA10;A:GLN36;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap13Native recall0.62
Jaccard0.54RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
3248 5.633988862191516 -0.911925 -23.9548 1 18 14 0.67 0.20 - no Open
2765 5.964406633404208 -0.633199 -15.3236 7 8 0 0.00 0.00 - no Open
2768 6.0638589157921725 -0.745837 -17.8865 4 10 0 0.00 0.00 - no Open
2767 6.774960579324483 -0.900122 -22.8247 6 12 0 0.00 0.00 - no Open
2766 5.888415266137783 -0.675755 -17.2578 2 9 0 0.00 0.00 - yes Open
2770 7.324050078057624 -0.781751 -19.979 4 16 0 0.00 0.00 - yes Open
3251 7.764661332364455 -0.944857 -23.0206 4 18 14 0.67 0.20 - yes Open
2769 8.107082940287334 -0.666123 -17.4904 6 10 0 0.00 0.00 - yes Open
3250 8.727101054323805 -0.933372 -22.5331 2 16 13 0.62 0.20 - yes Current
3249 9.010627289053046 -0.91508 -23.2618 1 17 14 0.67 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.533kcal/mol
Ligand efficiency (LE) -0.8667kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.985
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 361.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.19
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 17.95kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 79.82kcal/mol
Minimised FF energy 61.87kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.