FAIRMol

Z49595914

Pose ID 3244 Compound 440 Pose 3244

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Acceptable LE (-0.300 kcal/mol/HA) ✓ Good fit quality (FQ -3.13) ✗ Very high strain energy (86.9 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-11.995
kcal/mol
LE
-0.300
kcal/mol/HA
Fit Quality
-3.13
FQ (Leeson)
HAC
40
heavy atoms
MW
600
Da
LogP
5.35
cLogP
Strain ΔE
86.9 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: good
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 86.9 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 2 Clashes 7 Severe clashes 0
Final rank10.92539016925786Score-11.9947
Inter norm-0.537128Intra norm0.23726
Top1000noExcludedno
Contacts19H-bonds2
Artifact reasongeometry warning; 19 clashes; 7 protein contact clashes; high strain Δ 102.5
ResiduesA:ALA10;A:ARG29;A:ASN65;A:ASP22;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap16Native recall0.76
Jaccard0.67RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2538 8.003083200344426 -0.666796 -30.8424 5 20 0 0.00 0.00 - no Open
2536 8.437437849622983 -0.556673 -25.6625 3 19 0 0.00 0.00 - no Open
3241 8.46520447055287 -0.532882 -20.8008 5 18 14 0.67 0.20 - no Open
3857 8.558213222643754 -0.721445 -29.1179 4 18 0 0.00 0.00 - no Open
2533 8.632065822882883 -0.561726 -16.4217 4 20 0 0.00 0.00 - no Open
2834 9.055137518484493 -0.363995 -15.8167 4 11 0 0.00 0.00 - no Open
2535 9.396798971624426 -0.562936 -18.7431 4 17 0 0.00 0.00 - no Open
3859 9.614270776832695 -0.603368 -25.8221 3 14 0 0.00 0.00 - no Open
2534 9.915457705189256 -0.514385 -20.6039 3 18 0 0.00 0.00 - no Open
3238 10.629196938473772 -0.660263 -24.0087 4 20 16 0.76 0.20 - no Open
3244 10.92539016925786 -0.537128 -11.9947 2 19 16 0.76 0.20 - no Current
2539 9.52815942786826 -0.552126 -17.2889 3 18 0 0.00 0.00 - yes Open
2532 9.615744126318003 -0.481673 -22.4657 5 15 0 0.00 0.00 - yes Open
2835 10.219254722759766 -0.437208 -15.5695 5 16 0 0.00 0.00 - yes Open
2839 11.28855669180593 -0.481317 -16.1264 7 12 0 0.00 0.00 - yes Open
2833 11.51776014409267 -0.394523 -12.7379 5 16 0 0.00 0.00 - yes Open
3237 11.696324638842984 -0.597916 -21.0649 4 21 17 0.81 0.20 - yes Open
3862 11.703470114068287 -0.388639 -9.63917 3 15 0 0.00 0.00 - yes Open
3858 11.714360369687443 -0.407095 -14.7117 5 14 0 0.00 0.00 - yes Open
3240 11.842094196723728 -0.556641 -22.8259 5 19 16 0.76 0.20 - yes Open
3863 11.964607781403943 -0.448127 -20.6623 2 13 0 0.00 0.00 - yes Open
2837 11.99639711123841 -0.423874 -7.74164 4 13 0 0.00 0.00 - yes Open
3242 12.524835891285438 -0.581925 -22.737 4 21 17 0.81 0.20 - yes Open
2832 12.907279260886336 -0.410404 -17.3483 5 13 0 0.00 0.00 - yes Open
3861 13.785493187763784 -0.594342 -26.8524 4 14 0 0.00 0.00 - yes Open
3860 13.880118234272192 -0.479914 -17.8501 3 13 0 0.00 0.00 - yes Open
2838 14.012486292481311 -0.452397 -21.4487 8 13 0 0.00 0.00 - yes Open
2836 14.457260165522928 -0.41526 -17.6637 5 12 0 0.00 0.00 - yes Open
3864 14.607407259107656 -0.527173 -21.8525 3 14 0 0.00 0.00 - yes Open
3243 15.093291639828413 -0.549478 -17.8469 6 18 11 0.52 0.40 - yes Open
2537 15.10055491919647 -0.50444 -13.9192 5 16 0 0.00 0.00 - yes Open
3239 17.985371068956585 -0.626506 -25.519 6 23 16 0.76 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -11.995kcal/mol
Ligand efficiency (LE) -0.2999kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -3.132
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 40HA

Physicochemical properties

Molecular weight 600.1Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.35
Lipinski: ≤ 5
Rotatable bonds 9

Conformational strain (MMFF94s)

Strain energy (ΔE) 86.93kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 160.99kcal/mol
Minimised FF energy 74.06kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.