FAIRMol

Z30879796

Pose ID 3229 Compound 60 Pose 3229

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.767 kcal/mol/HA) ✓ Good fit quality (FQ -7.54) ✓ Good H-bonds (5 bonds) ✗ High strain energy (18.6 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-24.545
kcal/mol
LE
-0.767
kcal/mol/HA
Fit Quality
-7.54
FQ (Leeson)
HAC
32
heavy atoms
MW
488
Da
LogP
5.33
cLogP
Strain ΔE
18.6 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 18.6 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 2 Clashes 12 Severe clashes 6
Final rank13.570828863592425Score-24.5451
Inter norm-0.810768Intra norm0.0437349
Top1000noExcludedyes
Contacts18H-bonds5
Artifact reasonexcluded; geometry warning; 17 clashes; 6 protein clashes; moderate strain Δ 18.7
ResiduesA:ALA10;A:ARG29;A:ASP22;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:SER60;A:THR137;A:TYR122;A:TYR34;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap14Native recall0.67
Jaccard0.56RMSD-
H-bond strict2Strict recall0.40
H-bond same residue+role2Role recall0.40
H-bond same residue2Residue recall0.40

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
3230 3.301735402323313 -0.778387 -24.837 1 19 17 0.81 0.00 - no Open
2525 4.252925159304765 -0.729757 -22.1104 4 18 0 0.00 0.00 - no Open
2526 4.633907261580477 -0.716792 -21.76 3 18 0 0.00 0.00 - no Open
3229 13.570828863592425 -0.810768 -24.5451 5 18 14 0.67 0.40 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.545kcal/mol
Ligand efficiency (LE) -0.7670kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.543
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 488.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.33
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 18.58kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 141.16kcal/mol
Minimised FF energy 122.58kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.