FAIRMol

Z49582732

Pose ID 3175 Compound 443 Pose 3175

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.584 kcal/mol/HA) ✓ Good fit quality (FQ -5.85) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (61.7 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-19.868
kcal/mol
LE
-0.584
kcal/mol/HA
Fit Quality
-5.85
FQ (Leeson)
HAC
34
heavy atoms
MW
481
Da
LogP
4.53
cLogP
Strain ΔE
61.7 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 61.7 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 3 Clashes 13 Severe clashes 4
Final rank14.759476767944397Score-19.8678
Inter norm-0.678912Intra norm0.0945634
Top1000noExcludedyes
Contacts17H-bonds3
Artifact reasonexcluded; geometry warning; 16 clashes; 4 protein clashes; high strain Δ 62.0
ResiduesA:ALA10;A:ARG29;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO26;A:PRO27;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap12Native recall0.57
Jaccard0.46RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
3178 8.561225452286191 -0.597946 -15.6921 4 19 17 0.81 0.40 - no Open
3181 9.178150742018827 -0.6968 -22.311 2 20 19 0.90 0.40 - no Open
3176 9.273427524404912 -0.730579 -13.7786 3 21 18 0.86 0.20 - no Open
2208 9.332053475094035 -0.736386 -19.1927 0 16 0 0.00 0.00 - no Open
2890 9.351777890041042 -0.684534 -18.706 7 18 0 0.00 0.00 - no Open
2884 9.695369144262646 -0.55047 -14.5265 9 16 0 0.00 0.00 - no Open
2330 10.075589793746309 -0.816482 -25.0979 11 14 0 0.00 0.00 - no Open
2171 10.34880812517319 -0.939239 -28.1464 11 15 0 0.00 0.00 - no Open
2174 10.544682831572473 -0.77176 -22.7559 6 11 0 0.00 0.00 - no Open
2326 9.179645142698693 -0.663474 -17.5578 8 15 0 0.00 0.00 - yes Open
2325 10.22054777738333 -0.717665 -21.9072 11 17 0 0.00 0.00 - yes Open
2329 10.580682134405247 -0.739363 -24.0846 9 15 0 0.00 0.00 - yes Open
2207 10.594814460347544 -0.556055 -6.93792 4 17 0 0.00 0.00 - yes Open
2328 10.648916877177417 -0.637867 -17.8702 8 14 0 0.00 0.00 - yes Open
2887 10.712734239227101 -0.636859 -18.0653 11 13 0 0.00 0.00 - yes Open
2210 10.97681039861124 -0.851627 -19.6831 4 16 0 0.00 0.00 - yes Open
3177 11.008975613395442 -0.668741 -20.0653 2 20 18 0.86 0.40 - yes Open
2331 11.017205893859852 -0.765682 -21.5174 10 17 0 0.00 0.00 - yes Open
2173 11.038656642582188 -0.789011 -28.5754 8 17 0 0.00 0.00 - yes Open
3183 11.16436584579619 -0.646548 -16.6086 3 18 15 0.71 0.20 - yes Open
2206 11.203053045338944 -0.735342 -14.6301 1 14 0 0.00 0.00 - yes Open
2211 11.59640554655577 -0.746348 -22.7449 3 17 0 0.00 0.00 - yes Open
2175 11.611438314020434 -0.778434 -17.8094 13 17 0 0.00 0.00 - yes Open
3182 11.635782916121967 -0.704824 -20.8652 3 19 18 0.86 0.20 - yes Open
3184 11.675325310296653 -0.602876 -11.5392 3 18 14 0.67 0.40 - yes Open
2169 11.796479552715045 -0.78653 -16.841 10 17 0 0.00 0.00 - yes Open
2168 11.805667118246944 -0.923673 -25.9456 9 16 0 0.00 0.00 - yes Open
2332 11.806130018933356 -0.711398 -19.8184 9 18 0 0.00 0.00 - yes Open
2888 11.866923259069576 -0.727557 -22.9649 10 14 0 0.00 0.00 - yes Open
2327 11.88393810217282 -0.75158 -20.667 10 17 0 0.00 0.00 - yes Open
2881 11.985767806692772 -0.688236 -20.3951 8 17 0 0.00 0.00 - yes Open
2170 12.024862324890075 -0.847577 -27.4326 7 15 0 0.00 0.00 - yes Open
2883 12.448929720311018 -0.63381 -20.5646 9 16 0 0.00 0.00 - yes Open
2886 12.883497375178285 -0.722445 -21.2426 11 18 0 0.00 0.00 - yes Open
2212 12.961329528483635 -0.749899 -18.6328 1 14 0 0.00 0.00 - yes Open
2882 13.1402612192278 -0.595169 -7.89714 7 18 0 0.00 0.00 - yes Open
2885 13.202474894798751 -0.68163 -22.734 9 17 0 0.00 0.00 - yes Open
2889 13.228627783853733 -0.760975 -21.4321 9 17 0 0.00 0.00 - yes Open
3180 13.337831595790384 -0.705517 -17.5048 6 16 12 0.57 0.20 - yes Open
2172 13.641360761219438 -0.910092 -28.0326 7 15 0 0.00 0.00 - yes Open
3179 13.78453648987174 -0.780503 -24.7605 3 18 13 0.62 0.20 - yes Open
3175 14.759476767944397 -0.678912 -19.8678 3 17 12 0.57 0.20 - yes Current
2209 15.542191551637483 -0.691434 -20.8054 4 16 0 0.00 0.00 - yes Open
2205 16.369266440136705 -0.589797 -8.40918 6 18 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -19.868kcal/mol
Ligand efficiency (LE) -0.5843kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.847
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 480.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.53
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 61.68kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 116.85kcal/mol
Minimised FF energy 55.17kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.