FAIRMol

Z45800144

Pose ID 30768 Compound 2434 Pose 2747

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.935 kcal/mol/HA) ✓ Good fit quality (FQ -8.12) ✓ Good H-bonds (3 bonds) ✗ High strain energy (12.2 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-20.566
kcal/mol
LE
-0.935
kcal/mol/HA
Fit Quality
-8.12
FQ (Leeson)
HAC
22
heavy atoms
MW
308
Da
LogP
3.18
cLogP
Strain ΔE
12.2 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 22 π–π 0 Clashes 8 Severe clashes 0
Final rank3.927650825543325Score-20.5655
Inter norm-0.993653Intra norm0.0588583
Top1000noExcludedno
Contacts11H-bonds3
Artifact reasongeometry warning; 10 clashes; 8 protein contact clashes; moderate strain Δ 14.0
ResiduesA:ARG342;A:CYS26;A:GLN341;A:GLU343;A:GLU348;A:LEU339;A:LEU350;A:LEU382;A:PRO340;A:PRO344;A:PRO373

Protein summary

398 residues
Protein targetT14Atoms6140
Residues398Chains1
Residue summaryVAL:592; LEU:513; LYS:484; ARG:432; PHE:420; ILE:418; ASP:349; THR:322; TYR:315; PRO:308; GLU:301; ALA:290; SER:253; GLY:217; ASN:210; GLN:170

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name1NJJContacts15
PoseOpen native poseH-bonds7
IFP residuesA:ARG22; A:ARG242; A:ARG337; A:ARG342; A:ASP243; A:ASP385; A:GLN341; A:GLU384; A:LEU25; A:LEU339; A:LEU382; A:PRO340; A:PRO344; A:SER282; A:THR241
Current overlap6Native recall0.40
Jaccard0.30RMSD-
H-bond strict1Strict recall0.17
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2747 3.927650825543325 -0.993653 -20.5655 3 11 6 0.40 0.20 - no Current
2746 4.5702575415015545 -0.961315 -19.4994 5 13 8 0.53 0.20 - no Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.566kcal/mol
Ligand efficiency (LE) -0.9348kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.116
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 22HA

Physicochemical properties

Molecular weight 308.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.18
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 12.19kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 54.51kcal/mol
Minimised FF energy 42.32kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.