FAIRMol

Z56784540

Pose ID 3069 Compound 262 Pose 3069

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.641 kcal/mol/HA) ✓ Good fit quality (FQ -6.42) ✗ Very high strain energy (30.5 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-21.811
kcal/mol
LE
-0.641
kcal/mol/HA
Fit Quality
-6.42
FQ (Leeson)
HAC
34
heavy atoms
MW
467
Da
LogP
5.71
cLogP
Strain ΔE
30.5 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 30.5 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 2 Clashes 15 Severe clashes 3
Final rank59.725427282701794Score-21.8112
Inter norm-0.731909Intra norm0.0904037
Top1000noExcludedyes
Contacts20H-bonds2
Artifact reasonexcluded; geometry warning; 11 clashes; 3 protein clashes
ResiduesA:ALA10;A:ARG29;A:ASN65;A:ASP22;A:GLY117;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap17Native recall0.81
Jaccard0.71RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2580 5.160709902713007 -0.590921 -17.8316 6 11 0 0.00 0.00 - no Open
3066 5.178476442857638 -0.714923 -26.2833 3 17 14 0.67 0.00 - no Open
3070 5.422202675628983 -0.696439 -24.3513 2 19 17 0.81 0.20 - no Open
2577 5.423417647618024 -0.531526 -16.5011 7 14 0 0.00 0.00 - no Open
3064 5.981179083474143 -0.88379 -28.1667 2 19 15 0.71 0.00 - yes Open
2582 6.589048505643092 -0.445477 -18.6025 5 10 0 0.00 0.00 - yes Open
3068 6.73386768128858 -0.833162 -32.6734 3 18 14 0.67 0.20 - yes Open
3067 7.110240345645158 -0.800863 -23.9591 1 15 12 0.57 0.00 - yes Open
2583 7.719990143543413 -0.495318 -17.3941 5 13 0 0.00 0.00 - yes Open
2584 8.09953557343121 -0.488068 -14.8372 4 11 0 0.00 0.00 - yes Open
3065 8.28395616304644 -0.785058 -20.3553 1 19 16 0.76 0.20 - yes Open
2578 9.227845278060908 -0.522937 -10.6139 6 9 0 0.00 0.00 - yes Open
2581 57.261206707921524 -0.510444 -17.0586 5 11 0 0.00 0.00 - yes Open
2579 57.882324305812524 -0.541258 -15.7998 7 12 0 0.00 0.00 - yes Open
3063 58.41910120950779 -0.709047 -20.2755 5 15 14 0.67 0.00 - yes Open
3069 59.725427282701794 -0.731909 -21.8112 2 20 17 0.81 0.20 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.811kcal/mol
Ligand efficiency (LE) -0.6415kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.419
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 466.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.71
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 30.52kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 98.14kcal/mol
Minimised FF energy 67.61kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.