FAIRMol

Z56071437

Pose ID 3044 Compound 124 Pose 3044

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.818 kcal/mol/HA) ✓ Good fit quality (FQ -7.97) ✗ Very high strain energy (28.1 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-25.370
kcal/mol
LE
-0.818
kcal/mol/HA
Fit Quality
-7.97
FQ (Leeson)
HAC
31
heavy atoms
MW
500
Da
LogP
5.50
cLogP
Strain ΔE
28.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 28.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 5 Severe clashes 0
Final rank4.167622120393544Score-25.3697
Inter norm-0.823917Intra norm0.0055405
Top1000noExcludedno
Contacts18H-bonds1
Artifact reasongeometry warning; 11 clashes; 5 protein contact clashes; high strain Δ 27.1
ResiduesA:ALA10;A:ARG29;A:ASN65;A:GLN36;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:THR137;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap16Native recall0.76
Jaccard0.70RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2300 2.975199293457856 -0.795059 -28.9903 1 19 0 0.00 0.00 - no Open
3042 4.072703977033648 -0.910836 -30.2227 2 20 17 0.81 0.40 - no Open
3044 4.167622120393544 -0.823917 -25.3697 1 18 16 0.76 0.20 - no Current
2403 4.357679872175534 -0.685104 -21.0742 4 10 0 0.00 0.00 - no Open
3710 4.430265866663566 -0.727157 -21.84 4 14 0 0.00 0.00 - no Open
2187 4.616422523988748 -0.750283 -26.2709 6 13 0 0.00 0.00 - no Open
2549 4.825437208171437 -0.642671 -23.6962 5 10 0 0.00 0.00 - no Open
2018 4.939329756217788 -1.04522 -37.461 7 17 0 0.00 0.00 - no Open
3043 4.977027617950462 -0.770072 -27.1949 1 20 16 0.76 0.20 - no Open
2401 5.406678525852967 -0.689693 -24.6956 3 8 0 0.00 0.00 - no Open
1846 5.656921740362672 -0.936859 -32.4435 7 12 0 0.00 0.00 - no Open
1845 7.140819470640418 -0.992852 -33.9409 8 13 0 0.00 0.00 - no Open
2302 5.3690098490596245 -0.741315 -23.5675 3 15 0 0.00 0.00 - yes Open
3709 5.54423829292957 -0.754262 -27.3292 4 16 0 0.00 0.00 - yes Open
2188 6.363719603077262 -0.739161 -25.0271 5 15 0 0.00 0.00 - yes Open
2550 6.476803507875923 -0.607289 -22.283 3 11 0 0.00 0.00 - yes Open
2017 6.5810355141227594 -1.10765 -37.5989 7 16 0 0.00 0.00 - yes Open
3711 7.839426744555876 -0.62985 -20.2381 1 11 0 0.00 0.00 - yes Open
2551 8.096988315137459 -0.638837 -21.1506 7 11 0 0.00 0.00 - yes Open
2019 8.320791027619784 -0.838933 -26.3305 5 14 0 0.00 0.00 - yes Open
2301 8.420651808228492 -0.7417 -26.2675 2 17 0 0.00 0.00 - yes Open
2402 8.43645946478735 -0.580544 -21.5996 2 15 0 0.00 0.00 - yes Open
1847 8.500167348157591 -0.898004 -27.8574 11 11 0 0.00 0.00 - yes Open
2186 9.508457596523543 -0.894636 -26.6402 9 16 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -25.370kcal/mol
Ligand efficiency (LE) -0.8184kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.973
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 31HA

Physicochemical properties

Molecular weight 500.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.50
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 28.12kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 46.14kcal/mol
Minimised FF energy 18.02kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.