FAIRMol

Z169788636

Pose ID 3038 Compound 55 Pose 3038

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.920 kcal/mol/HA) ✓ Good fit quality (FQ -8.36) ✗ High strain energy (14.2 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-22.990
kcal/mol
LE
-0.920
kcal/mol/HA
Fit Quality
-8.36
FQ (Leeson)
HAC
25
heavy atoms
MW
333
Da
LogP
2.66
cLogP
Strain ΔE
14.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 14.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 1 Clashes 4 Severe clashes 0
Final rank3.2235175485160297Score-22.9897
Inter norm-0.947757Intra norm0.0281671
Top1000noExcludedno
Contacts17H-bonds2
Artifact reasongeometry warning; 12 clashes; 4 protein contact clashes; moderate strain Δ 18.9
ResiduesA:ALA10;A:ASN65;A:GLU31;A:GLY117;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap17Native recall0.81
Jaccard0.81RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2162 2.9229996401785945 -0.963315 -23.4056 3 17 0 0.00 0.00 - no Open
3038 3.2235175485160297 -0.947757 -22.9897 2 17 17 0.81 0.20 - no Current
3040 3.5342847236341126 -0.974722 -24.7949 2 16 16 0.76 0.20 - no Open
2279 4.309629141589049 -1.01231 -24.6167 2 17 0 0.00 0.00 - no Open
2277 4.5141769966606615 -0.954387 -24.2737 1 18 0 0.00 0.00 - no Open
3039 4.889083601580632 -0.982322 -21.5005 2 14 10 0.48 0.20 - yes Open
3041 5.371919715087432 -0.881115 -18.7058 1 16 16 0.76 0.20 - yes Open
2278 6.8513170825807705 -0.964752 -20.2175 2 14 0 0.00 0.00 - yes Open
2280 7.769774725740086 -1.10015 -26.0693 2 16 0 0.00 0.00 - yes Open
2163 8.836912964051276 -1.01737 -22.0739 5 15 0 0.00 0.00 - yes Open
2164 9.412729799491025 -1.06641 -24.4858 5 15 0 0.00 0.00 - yes Open
2165 11.056390803496809 -1.10482 -21.3976 7 15 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.990kcal/mol
Ligand efficiency (LE) -0.9196kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.360
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 25HA

Physicochemical properties

Molecular weight 333.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.66
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 14.15kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 12.47kcal/mol
Minimised FF energy -1.69kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.