FAIRMol

Z56891526

Pose ID 30239 Compound 2349 Pose 2218

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.198 kcal/mol/HA) ✓ Good fit quality (FQ -9.82) ✓ Strong H-bond network (8 bonds) ✗ High strain energy (12.4 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-22.762
kcal/mol
LE
-1.198
kcal/mol/HA
Fit Quality
-9.82
FQ (Leeson)
HAC
19
heavy atoms
MW
280
Da
LogP
-0.53
cLogP
Strain ΔE
12.4 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 8 Hydrophobic 0 π–π 0 Clashes 4 Severe clashes 0 ⚠ Hydrophobic exposure 100%
🚨Solvent-exposed hydrophobic surface — desolvation penalty likely
100% of hydrophobic surface is solvent-exposed (12/12 atoms). Large non-polar area without protein contacts incurs a desolvation penalty and will reduce binding affinity. Consider truncating or replacing the exposed fragment.
Non-polar atoms 12 Buried (contacted) 0 Exposed 12 LogP -0.53 H-bonds 8
Exposed fragments: phenyl (3/5 atoms exposed)phenyl (6/6 atoms exposed)aliphatic chain/group (3 atoms exposed)
Final rank2.026871902667413Score-22.7618
Inter norm-1.14291Intra norm-0.0550831
Top1000noExcludedno
Contacts8H-bonds8
Artifact reasongeometry warning; 4 clashes; 4 protein contact clashes; high strain Δ 22.3
ResiduesA:ARG337;A:ASP243;A:ASP385;A:GLU384;A:LEU339;A:MET386;A:PHE383;A:VAL336

Protein summary

398 residues
Protein targetT14Atoms6140
Residues398Chains1
Residue summaryVAL:592; LEU:513; LYS:484; ARG:432; PHE:420; ILE:418; ASP:349; THR:322; TYR:315; PRO:308; GLU:301; ALA:290; SER:253; GLY:217; ASN:210; GLN:170

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name1NJJContacts15
PoseOpen native poseH-bonds7
IFP residuesA:ARG22; A:ARG242; A:ARG337; A:ARG342; A:ASP243; A:ASP385; A:GLN341; A:GLU384; A:LEU25; A:LEU339; A:LEU382; A:PRO340; A:PRO344; A:SER282; A:THR241
Current overlap5Native recall0.33
Jaccard0.28RMSD-
H-bond strict1Strict recall0.17
H-bond same residue+role2Role recall0.40
H-bond same residue2Residue recall0.40

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

No hydrophobic contacts detected for this pose.

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2218 2.026871902667413 -1.14291 -22.7618 8 8 5 0.33 0.40 - no Current
2240 2.6603027078915193 -1.13227 -21.2646 10 9 7 0.47 0.40 - no Open
2225 2.926559441366489 -0.984292 -18.1629 6 8 5 0.33 0.20 - no Open
2244 2.9994837867102038 -1.06455 -18.2589 7 9 7 0.47 0.20 - no Open
2033 3.005426615928177 -1.10122 -24.3358 6 13 0 0.00 0.00 - no Open
2233 3.0305860436455854 -0.967732 -18.5018 6 10 7 0.47 0.20 - no Open
2031 3.439757743207278 -1.23837 -22.0394 7 15 0 0.00 0.00 - no Open
2219 3.6736360702498603 -1.23432 -16.3059 8 11 7 0.47 0.20 - no Open
2232 3.7109895108672033 -1.38009 -23.3596 8 10 7 0.47 0.20 - no Open
2239 3.7301979323386565 -1.16731 -21.1186 10 11 8 0.53 0.40 - no Open
2224 3.8131917456090445 -1.31688 -21.5211 8 10 7 0.47 0.40 - no Open
2006 3.938484542984906 -1.47514 -23.7311 7 14 0 0.00 0.00 - no Open
2241 4.0573841509592175 -0.956382 -19.1841 6 11 5 0.33 0.20 - no Open
2009 3.64336835867456 -1.23336 -23.2299 7 14 0 0.00 0.00 - yes Open
2023 3.8576950139824273 -1.28078 -22.0359 6 14 0 0.00 0.00 - yes Open
2217 3.8614512475870413 -1.25539 -20.7896 6 9 5 0.33 0.20 - yes Open
2015 4.045196438237178 -1.26347 -21.3339 7 15 0 0.00 0.00 - yes Open
2235 4.061172695494321 -0.908576 -12.0235 5 9 7 0.47 0.20 - yes Open
2229 4.184803569541945 -1.2042 -21.0722 5 10 5 0.33 0.20 - yes Open
2035 4.490157721600345 -1.12032 -18.8623 7 14 0 0.00 0.00 - yes Open
2221 4.518052043509275 -1.38391 -21.9055 7 10 6 0.40 0.20 - yes Open
2236 4.702686246712027 -0.995458 -20.7366 7 11 8 0.53 0.60 - yes Open
2029 4.803072175671976 -1.12471 -19.6841 8 14 0 0.00 0.00 - yes Open
2013 4.866254858817714 -1.33469 -23.7553 7 15 0 0.00 0.00 - yes Open
2222 4.868191230149295 -1.1976 -22.6408 11 9 5 0.33 0.20 - yes Open
2223 4.915543641676009 -1.44788 -26.1058 7 10 8 0.53 0.40 - yes Open
2017 5.1515721798021765 -1.10403 -18.7275 7 14 0 0.00 0.00 - yes Open
2032 5.328442844841178 -1.14634 -22.1108 8 15 0 0.00 0.00 - yes Open
2238 5.40584278815577 -1.03792 -20.3077 9 11 6 0.40 0.20 - yes Open
2230 5.68916261214194 -1.31052 -24.1428 8 11 6 0.40 0.20 - yes Open
2024 5.761255144045803 -1.27891 -19.7006 8 14 0 0.00 0.00 - yes Open
2215 5.782772674582591 -1.44079 -25.3918 7 10 8 0.53 0.40 - yes Open
2246 5.823329495083621 -1.36096 -24.4997 10 11 6 0.40 0.20 - yes Open
2019 5.890182783520056 -1.3051 -17.7785 7 17 0 0.00 0.00 - yes Open
2037 5.894511591378404 -1.12067 -21.8113 7 12 0 0.00 0.00 - yes Open
2025 5.978723121372389 -1.06654 -22.662 6 14 0 0.00 0.00 - yes Open
2026 6.002792951217877 -1.37637 -24.056 11 14 0 0.00 0.00 - yes Open
2245 6.085644639233802 -0.996695 -16.3884 5 10 6 0.40 0.20 - yes Open
2016 6.118152948823159 -1.09185 -18.5692 8 14 0 0.00 0.00 - yes Open
2012 6.125664527902213 -1.27859 -20.6399 8 15 0 0.00 0.00 - yes Open
2234 6.147505467060259 -1.11666 -20.1522 5 10 6 0.40 0.20 - yes Open
2027 6.282088696229935 -1.24298 -22.9085 8 13 0 0.00 0.00 - yes Open
2010 6.3285950573094745 -1.53038 -22.5993 10 16 0 0.00 0.00 - yes Open
2007 6.375508283178409 -1.36617 -21.9488 8 14 0 0.00 0.00 - yes Open
2227 6.442677896213871 -1.26053 -20.4678 7 12 6 0.40 0.40 - yes Open
2036 6.541446118972117 -1.21648 -20.0421 7 12 0 0.00 0.00 - yes Open
2018 7.3119849345106305 -1.27495 -21.1875 7 16 0 0.00 0.00 - yes Open
2021 7.602828333694626 -1.14254 -22.8145 8 12 0 0.00 0.00 - yes Open
2226 54.35881857057994 -1.14038 -20.5263 6 10 6 0.40 0.20 - yes Open
2008 54.84243709664221 -1.39776 -22.4524 8 15 0 0.00 0.00 - yes Open
2231 55.099938857539584 -1.30828 -20.4055 6 9 7 0.47 0.20 - yes Open
2030 55.374439016037485 -1.3945 -25.7136 8 15 0 0.00 0.00 - yes Open
2228 55.66950002303142 -1.13288 -18.9641 7 8 5 0.33 0.20 - yes Open
2011 55.71464406906111 -1.45556 -25.2589 8 13 0 0.00 0.00 - yes Open
2028 55.82138655876557 -1.16562 -19.7479 8 16 0 0.00 0.00 - yes Open
2220 55.86528566775287 -1.30055 -22.6264 7 10 7 0.47 0.20 - yes Open
2022 55.95191748638111 -1.40855 -23.5316 12 16 0 0.00 0.00 - yes Open
2242 55.974407454042655 -1.11278 -22.2904 5 11 6 0.40 0.20 - yes Open
2034 56.21764766101079 -1.25071 -14.3425 12 17 0 0.00 0.00 - yes Open
2014 56.30159903302769 -1.34144 -24.6298 11 15 0 0.00 0.00 - yes Open
2237 56.43784972685953 -1.08522 -18.4297 8 11 7 0.47 0.20 - yes Open
2216 56.58339452851141 -1.25857 -20.7031 8 11 6 0.40 0.20 - yes Open
2243 56.702632901700554 -1.02299 -16.3893 7 9 5 0.33 0.20 - yes Open
2020 57.45909968129073 -1.14936 -20.3795 6 13 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.762kcal/mol
Ligand efficiency (LE) -1.1980kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.820
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 19HA

Physicochemical properties

Molecular weight 280.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) -0.53
Lipinski: ≤ 5
Rotatable bonds 2

Conformational strain (MMFF94s)

Strain energy (ΔE) 12.42kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 83.88kcal/mol
Minimised FF energy 71.46kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.