FAIRMol

Z56905026

Pose ID 2994 Compound 36 Pose 2994

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.798 kcal/mol/HA) ✓ Good fit quality (FQ -7.35) ✓ Good H-bonds (4 bonds) ✗ Very high strain energy (29.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-20.749
kcal/mol
LE
-0.798
kcal/mol/HA
Fit Quality
-7.35
FQ (Leeson)
HAC
26
heavy atoms
MW
375
Da
LogP
2.36
cLogP
Strain ΔE
29.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: mixed
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 29.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 18 π–π 0 Clashes 8 Severe clashes 2
Final rank7.346863824897405Score-20.749
Inter norm-0.805001Intra norm0.00696126
Top1000noExcludedyes
Contacts16H-bonds4
Artifact reasonexcluded; geometry warning; 5 clashes; 2 protein clashes; high strain Δ 42.9
ResiduesA:ALA10;A:ARG29;A:GLU31;A:ILE139;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:THR137;A:TRP25;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap11Native recall0.52
Jaccard0.42RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2991 2.997113147971836 -0.767833 -22.0119 3 17 17 0.81 0.00 - no Open
2987 3.444094259103178 -0.751584 -22.4756 4 17 16 0.76 0.00 - no Open
2988 3.9824329765574076 -0.97239 -17.1657 4 19 15 0.71 0.20 - no Open
2998 4.59751239423209 -0.707089 -15.6032 5 15 12 0.57 0.20 - no Open
3007 5.4529768270059655 -0.831001 -17.1903 5 17 14 0.67 0.20 - no Open
3005 5.792279709509073 -0.964176 -25.0979 5 16 12 0.57 0.20 - no Open
3525 6.080960831117881 -0.729444 -18.8085 5 14 0 0.00 0.00 - no Open
3528 6.082201155027588 -0.746597 -21.5305 8 13 0 0.00 0.00 - no Open
2993 5.230362432030884 -1.03804 -25.3916 5 21 16 0.76 0.20 - yes Open
3526 5.343907756949862 -0.788933 -22.2437 10 13 0 0.00 0.00 - yes Open
3006 5.382400922174863 -0.826328 -24.226 6 16 16 0.76 0.40 - yes Open
3010 5.539793732392567 -0.783476 -22.5256 2 15 14 0.67 0.00 - yes Open
3523 5.661532641631642 -0.676736 -26.8993 7 13 0 0.00 0.00 - yes Open
3519 5.6714789893344575 -0.663428 -19.828 5 14 0 0.00 0.00 - yes Open
3011 5.799051701768517 -0.642957 -19.2261 2 18 18 0.86 0.20 - yes Open
3522 5.804360078828302 -0.75195 -17.6548 10 13 0 0.00 0.00 - yes Open
2995 5.941132940468755 -0.712507 -16.501 4 16 16 0.76 0.20 - yes Open
3527 5.984808635547948 -0.705539 -20.3691 5 13 0 0.00 0.00 - yes Open
3002 6.134372114881237 -0.740427 -24.3675 1 14 13 0.62 0.00 - yes Open
3001 6.588051363059027 -1.01094 -24.6974 5 18 14 0.67 0.20 - yes Open
2999 7.096869829155203 -0.72471 -18.8892 5 14 14 0.67 0.20 - yes Open
3000 7.184326804783248 -0.988801 -31.2802 5 17 13 0.62 0.20 - yes Open
2994 7.346863824897405 -0.805001 -20.749 4 16 11 0.52 0.20 - yes Current
2985 7.386093357325582 -1.0232 -27.3526 5 17 12 0.57 0.20 - yes Open
3520 7.402849849892192 -0.800402 -20.1911 6 10 0 0.00 0.00 - yes Open
3518 7.620015898578951 -0.891711 -25.1924 6 15 0 0.00 0.00 - yes Open
2997 8.581906008119264 -0.970149 -23.419 5 19 15 0.71 0.20 - yes Open
2989 8.710329391784898 -1.09795 -24.8055 8 20 13 0.62 0.20 - yes Open
3009 10.059422149524359 -0.924697 -24.2246 5 19 15 0.71 0.20 - yes Open
2984 11.390057096671027 -0.928895 -23.5751 5 20 14 0.67 0.20 - yes Open
3524 55.52690077775039 -0.861394 -20.1102 7 12 0 0.00 0.00 - yes Open
2992 57.11387945491687 -1.02653 -26.1732 5 19 14 0.67 0.20 - yes Open
3529 57.46898647201772 -0.697004 -18.9309 5 16 0 0.00 0.00 - yes Open
3004 57.68315125019384 -0.915303 -16.1836 6 19 15 0.71 0.40 - yes Open
3521 57.85908129187729 -1.00856 -24.0747 8 13 0 0.00 0.00 - yes Open
2996 58.35508053203513 -0.988933 -22.4372 5 20 15 0.71 0.20 - yes Open
3008 58.41002135179489 -1.03562 -23.8992 5 19 14 0.67 0.20 - yes Open
3003 58.4167327681313 -0.648384 -16.198 6 17 16 0.76 0.40 - yes Open
2990 60.243407219128166 -0.919276 -15.9649 5 16 11 0.52 0.20 - yes Open
2986 60.46007970472873 -0.808032 -20.5762 6 17 12 0.57 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.749kcal/mol
Ligand efficiency (LE) -0.7980kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.353
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 375.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.36
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 29.41kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 107.93kcal/mol
Minimised FF energy 78.53kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.