FAIRMol

Z49620424

Pose ID 2969 Compound 277 Pose 2969

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.577 kcal/mol/HA) ✓ Good fit quality (FQ -5.32) ✗ Very high strain energy (34.0 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-15.008
kcal/mol
LE
-0.577
kcal/mol/HA
Fit Quality
-5.32
FQ (Leeson)
HAC
26
heavy atoms
MW
344
Da
LogP
3.80
cLogP
Strain ΔE
34.0 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 34.0 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 4 Severe clashes 1
Final rank5.4826108951854104Score-15.008
Inter norm-0.799545Intra norm0.222313
Top1000noExcludedyes
Contacts19H-bonds1
Artifact reasonexcluded; geometry warning; 10 clashes; 1 protein clash; high strain Δ 34.3
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLN36;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.82RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2895 3.5680366603155624 -0.875622 -17.9281 2 16 0 0.00 0.00 - no Open
2899 4.248941167689489 -0.859109 -17.5979 2 16 0 0.00 0.00 - no Open
2965 5.308998017938502 -0.823275 -13.2672 4 14 14 0.67 0.00 - no Open
2897 5.4955598640357195 -0.961178 -32.5747 4 16 0 0.00 0.00 - no Open
1977 6.128192467707609 -0.669275 -12.3648 5 13 0 0.00 0.00 - no Open
2972 6.194229119201112 -0.759884 -24.8264 4 16 16 0.76 0.40 - no Open
2969 5.4826108951854104 -0.799545 -15.008 1 19 18 0.86 0.00 - yes Current
1983 5.48304453668463 -0.748913 -23.2812 3 11 0 0.00 0.00 - yes Open
2975 5.793326680599963 -0.867062 -27.5297 5 16 16 0.76 0.00 - yes Open
2966 6.279142669862784 -0.920731 -17.9824 4 15 13 0.62 0.00 - yes Open
2893 6.4666777375179905 -1.05125 -32.6316 5 18 0 0.00 0.00 - yes Open
2901 6.8441236080302135 -0.946837 -29.7856 4 16 0 0.00 0.00 - yes Open
2891 6.899870697519042 -0.969732 -18.8968 3 16 0 0.00 0.00 - yes Open
1975 7.352614391475464 -0.783317 -24.7821 3 13 0 0.00 0.00 - yes Open
2973 7.556308040680262 -0.807806 -13.1415 4 18 17 0.81 0.20 - yes Open
1979 7.585627526526178 -0.875149 -29.1481 3 12 0 0.00 0.00 - yes Open
1981 7.701763351511589 -0.795936 -15.9514 4 18 0 0.00 0.00 - yes Open
2964 7.886850331576594 -0.854572 -16.2031 4 18 18 0.86 0.00 - yes Open
2970 8.536235146237935 -0.896245 -18.7475 5 19 16 0.76 0.20 - yes Open
1978 8.644023613410653 -0.790913 -22.6078 3 12 0 0.00 0.00 - yes Open
2900 8.725908158089055 -0.844865 -19.9325 4 7 0 0.00 0.00 - yes Open
2971 8.82514382914119 -0.914161 -29.0172 5 16 16 0.76 0.00 - yes Open
1982 9.556985410314299 -0.708518 -26.3645 2 11 0 0.00 0.00 - yes Open
1973 9.746988212221206 -1.00647 -17.7989 7 18 0 0.00 0.00 - yes Open
1972 10.613239270658962 -0.873823 -24.9601 7 17 0 0.00 0.00 - yes Open
2892 10.842537185624233 -1.02671 -24.4977 5 10 0 0.00 0.00 - yes Open
2894 11.600767925025217 -0.855338 -26.0604 3 15 0 0.00 0.00 - yes Open
2967 58.26173349716666 -0.983468 -27.7945 5 17 16 0.76 0.00 - yes Open
2898 58.58646118643031 -0.848977 -17.4653 3 11 0 0.00 0.00 - yes Open
1976 59.49070500352732 -0.653322 -21.0698 2 12 0 0.00 0.00 - yes Open
2968 60.1173914487811 -0.739205 -22.7182 4 17 15 0.71 0.00 - yes Open
2974 60.53293236544626 -0.803751 -23.9808 5 15 12 0.57 0.20 - yes Open
1974 61.18086007502781 -0.864941 -27.6485 6 12 0 0.00 0.00 - yes Open
2896 61.4266105010899 -1.03491 -31.8934 8 11 0 0.00 0.00 - yes Open
1980 61.8958568934499 -0.746372 -20.1676 4 12 0 0.00 0.00 - yes Open
2890 62.56409004457617 -0.939617 -27.9805 4 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -15.008kcal/mol
Ligand efficiency (LE) -0.5772kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.318
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 344.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.80
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 34.03kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 124.01kcal/mol
Minimised FF energy 89.98kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.