FAIRMol

ulfkktlib_2370

Pose ID 28882 Compound 2391 Pose 861

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-2.183 kcal/mol/HA) ✓ Good fit quality (FQ -13.07) ✓ Strong H-bond network (10 bonds) ✗ Moderate strain (7.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-21.834
kcal/mol
LE
-2.183
kcal/mol/HA
Fit Quality
-13.07
FQ (Leeson)
HAC
10
heavy atoms
MW
205
Da
LogP
-0.18
cLogP
Strain ΔE
7.0 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 10 Hydrophobic 1 π–π 0 Clashes 7 Severe clashes 0 ⚠ Hydrophobic exposure 100%
🚨Solvent-exposed hydrophobic surface — desolvation penalty likely
100% of hydrophobic surface is solvent-exposed (4/4 atoms). Large non-polar area without protein contacts incurs a desolvation penalty and will reduce binding affinity. Consider truncating or replacing the exposed fragment.
Non-polar atoms 4 Buried (contacted) 0 Exposed 4 LogP -0.18 H-bonds 10
Exposed fragments: aromatic ring (4/6 atoms exposed)
Final rank1.3286563099559354Score-21.8338
Inter norm-2.21009Intra norm0.0267192
Top1000noExcludedno
Contacts9H-bonds10
Artifact reasongeometry warning; 4 clashes; 7 protein contact clashes; moderate strain Δ 15.8
ResiduesA:ARG337;A:ASP243;A:ASP385;A:GLU384;A:LEU339;A:MET386;A:PHE383;A:PRO338;A:VAL336

Protein summary

398 residues
Protein targetT14Atoms6140
Residues398Chains1
Residue summaryVAL:592; LEU:513; LYS:484; ARG:432; PHE:420; ILE:418; ASP:349; THR:322; TYR:315; PRO:308; GLU:301; ALA:290; SER:253; GLY:217; ASN:210; GLN:170

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name1NJJContacts15
PoseOpen native poseH-bonds7
IFP residuesA:ARG22; A:ARG242; A:ARG337; A:ARG342; A:ASP243; A:ASP385; A:GLN341; A:GLU384; A:LEU25; A:LEU339; A:LEU382; A:PRO340; A:PRO344; A:SER282; A:THR241
Current overlap5Native recall0.33
Jaccard0.26RMSD-
H-bond strict2Strict recall0.33
H-bond same residue+role3Role recall0.60
H-bond same residue3Residue recall0.60

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
861 1.3286563099559354 -2.21009 -21.8338 10 9 5 0.33 0.60 - no Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.834kcal/mol
Ligand efficiency (LE) -2.1834kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -13.074
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 10HA

Physicochemical properties

Molecular weight 205.0Da
Lipinski: ≤ 500 Da
LogP (cLogP) -0.18
Lipinski: ≤ 5
Rotatable bonds 1

Conformational strain (MMFF94s)

Strain energy (ΔE) 7.00kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 53.13kcal/mol
Minimised FF energy 46.13kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.