FAIRMol

Z48204477

Pose ID 2887 Compound 211 Pose 2887

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.682 kcal/mol/HA) ✓ Good fit quality (FQ -6.93) ✗ High strain energy (15.5 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-24.538
kcal/mol
LE
-0.682
kcal/mol/HA
Fit Quality
-6.93
FQ (Leeson)
HAC
36
heavy atoms
MW
491
Da
LogP
4.09
cLogP
Strain ΔE
15.5 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 15.5 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 3 Clashes 5 Severe clashes 1
Final rank5.224116412819443Score-24.5382
Inter norm-0.665305Intra norm-0.0163119
Top1000noExcludedyes
Contacts16H-bonds1
Artifact reasonexcluded; geometry warning; 13 clashes; 1 protein clash; moderate strain Δ 15.7
ResiduesA:ALA10;A:ARG29;A:ASP22;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap14Native recall0.67
Jaccard0.61RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2885 4.723822499803568 -0.697344 -25.1592 1 16 16 0.76 0.20 - no Open
2887 5.224116412819443 -0.665305 -24.5382 1 16 14 0.67 0.00 - yes Current
2888 8.282901503495166 -0.581127 -16.7701 0 18 15 0.71 0.00 - yes Open
2886 58.3282136248833 -0.654389 -23.583 1 18 14 0.67 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.538kcal/mol
Ligand efficiency (LE) -0.6816kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.928
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 36HA

Physicochemical properties

Molecular weight 490.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.09
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 15.46kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 98.40kcal/mol
Minimised FF energy 82.94kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.