FAIRMol

Z44851564

Pose ID 2876 Compound 27 Pose 2876

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.878 kcal/mol/HA) ✓ Good fit quality (FQ -7.75) ✗ High strain energy (11.5 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-20.191
kcal/mol
LE
-0.878
kcal/mol/HA
Fit Quality
-7.75
FQ (Leeson)
HAC
23
heavy atoms
MW
301
Da
LogP
3.87
cLogP
Strain ΔE
11.5 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 1 Clashes 5 Severe clashes 0
Final rank2.8319733988319324Score-20.1913
Inter norm-1.07994Intra norm0.202064
Top1000noExcludedno
Contacts15H-bonds2
Artifact reasongeometry warning; 10 clashes; 5 protein contact clashes; moderate strain Δ 12.2
ResiduesA:ALA10;A:ASN65;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap15Native recall0.71
Jaccard0.71RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2877 2.737543921059323 -1.04073 -19.2706 1 15 15 0.71 0.20 - no Open
2876 2.8319733988319324 -1.07994 -20.1913 2 15 15 0.71 0.00 - no Current
2879 3.114708662724084 -1.06929 -20.2654 1 16 16 0.76 0.20 - no Open
2880 3.4316045754720603 -1.00264 -21.8981 0 14 14 0.67 0.00 - no Open
2875 3.8368808687190947 -1.05499 -25.0674 1 16 16 0.76 0.20 - no Open
2878 4.161187415348698 -0.9905 -21.6566 2 14 11 0.52 0.20 - no Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.191kcal/mol
Ligand efficiency (LE) -0.8779kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.748
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 23HA

Physicochemical properties

Molecular weight 301.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.87
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 11.54kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 103.63kcal/mol
Minimised FF energy 92.09kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.