FAIRMol

Z57045660

Pose ID 2842 Compound 290 Pose 2842

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.605 kcal/mol/HA) ✓ Good fit quality (FQ -6.05) ✗ Very high strain energy (33.3 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-20.553
kcal/mol
LE
-0.605
kcal/mol/HA
Fit Quality
-6.05
FQ (Leeson)
HAC
34
heavy atoms
MW
498
Da
LogP
3.87
cLogP
Strain ΔE
33.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 33.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 4 Severe clashes 1
Final rank6.309150452737945Score-20.5534
Inter norm-0.503854Intra norm-0.100657
Top1000noExcludedyes
Contacts19H-bonds1
Artifact reasonexcluded; geometry warning; 12 clashes; 1 protein clash; high strain Δ 39.2
ResiduesA:ALA10;A:ARG29;A:ASN65;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:THR137;A:THR57;A:TYR122;A:TYR34;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap16Native recall0.76
Jaccard0.67RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2843 5.37493306530174 -0.591587 -19.5559 1 19 19 0.90 0.00 - no Open
2842 6.309150452737945 -0.503854 -20.5534 1 19 16 0.76 0.20 - yes Current
2841 6.695718809532638 -0.723743 -24.1493 3 19 18 0.86 0.20 - yes Open
2840 55.771118069546716 -0.619649 -20.4988 1 19 18 0.86 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.553kcal/mol
Ligand efficiency (LE) -0.6045kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.049
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 498.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.87
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 33.31kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 104.07kcal/mol
Minimised FF energy 70.77kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.