FAIRMol

Z56911531

Pose ID 2718 Compound 2 Pose 2718

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.922 kcal/mol/HA) ✓ Good fit quality (FQ -8.13) ✗ Very high strain energy (26.2 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-21.197
kcal/mol
LE
-0.922
kcal/mol/HA
Fit Quality
-8.13
FQ (Leeson)
HAC
23
heavy atoms
MW
348
Da
LogP
0.89
cLogP
Strain ΔE
26.2 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 20 π–π 2 Clashes 3 Severe clashes 0
Final rank2.8147308630186267Score-21.1968
Inter norm-0.988936Intra norm0.0673367
Top1000noExcludedno
Contacts18H-bonds2
Artifact reasongeometry warning; 5 clashes; 3 protein contact clashes; high strain Δ 32.7
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLN36;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.86RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2723 1.5604197035524388 -0.913775 -22.2171 1 17 17 0.81 0.00 - no Open
2029 1.7059713643461074 -0.837053 -23.0529 5 8 0 0.00 0.00 - no Open
2735 2.3111223783425956 -0.982622 -22.4013 2 16 16 0.76 0.00 - no Open
2719 2.443999222667504 -1.08329 -28.6246 3 15 15 0.71 0.00 - no Open
2731 2.5119241442476508 -0.935561 -19.97 3 16 16 0.76 0.00 - no Open
2041 2.5439755131995523 -0.740474 -21.248 5 9 0 0.00 0.00 - no Open
2711 2.7208662803081243 -1.09767 -28.3151 3 16 16 0.76 0.00 - no Open
2727 2.7595859848853452 -0.974629 -23.1355 3 15 15 0.71 0.00 - no Open
2718 2.8147308630186267 -0.988936 -21.1968 2 18 18 0.86 0.00 - no Current
2032 2.8224908567566755 -0.8561 -21.5287 5 9 0 0.00 0.00 - no Open
2033 2.8830022927260677 -0.693302 -17.6633 3 11 0 0.00 0.00 - no Open
2710 3.029289646652832 -0.968187 -19.9388 1 17 17 0.81 0.00 - no Open
2722 3.0405012201603463 -0.899559 -18.7293 2 16 16 0.76 0.00 - no Open
2737 3.0528231105701473 -1.16313 -27.565 7 15 11 0.52 0.20 - no Open
2036 3.2718526512040342 -0.577733 -15.9609 4 8 0 0.00 0.00 - no Open
2030 3.455771088204806 -0.788762 -18.9118 7 13 0 0.00 0.00 - no Open
2715 3.4672852949471844 -0.986468 -22.6932 3 14 14 0.67 0.00 - no Open
2037 3.545850608455604 -0.682465 -18.9718 4 9 0 0.00 0.00 - no Open
2028 3.6055367436199335 -0.9424 -21.5142 6 8 0 0.00 0.00 - no Open
2039 3.629856557472742 -0.699599 -13.3474 3 7 0 0.00 0.00 - no Open
2035 3.6957795670297346 -0.686793 -14.8885 5 10 0 0.00 0.00 - no Open
2027 4.324578345788533 -0.718888 -17.846 4 8 0 0.00 0.00 - no Open
2714 3.440963953338777 -0.944613 -21.5359 3 18 18 0.86 0.00 - yes Open
2734 3.6230834723422647 -0.966563 -20.9662 1 17 17 0.81 0.00 - yes Open
2739 4.140794520963718 -0.93285 -22.1859 4 14 14 0.67 0.00 - yes Open
2040 4.198066759162342 -0.73896 -14.4806 8 12 0 0.00 0.00 - yes Open
2726 5.244296371748054 -1.03678 -25.2534 3 15 15 0.71 0.00 - yes Open
2721 5.484065974017065 -1.18397 -25.2273 5 16 12 0.57 0.20 - yes Open
2736 5.85566946690933 -1.20895 -29.0923 5 17 13 0.62 0.20 - yes Open
2716 6.169568233495898 -1.18321 -26.0767 5 17 12 0.57 0.20 - yes Open
2708 6.353841363669128 -1.22504 -24.9577 6 18 13 0.62 0.20 - yes Open
2728 6.6765937669926085 -1.15455 -28.6266 6 17 13 0.62 0.20 - yes Open
2729 6.971296429575896 -1.07441 -24.8012 8 19 14 0.67 0.20 - yes Open
2724 7.882734148557311 -1.18142 -25.8765 5 20 15 0.71 0.20 - yes Open
2712 7.927944404961771 -1.17532 -26.4727 6 18 13 0.62 0.20 - yes Open
2732 8.355355084833475 -1.1045 -24.7218 4 16 12 0.57 0.20 - yes Open
2034 53.10310312177632 -0.760402 -16.8035 4 7 0 0.00 0.00 - yes Open
2038 54.8401540411849 -0.702908 -20.8888 2 7 0 0.00 0.00 - yes Open
2031 55.13596661923141 -0.784891 -15.483 2 13 0 0.00 0.00 - yes Open
2709 56.102615384697685 -1.18289 -24.5438 6 16 13 0.62 0.20 - yes Open
2720 56.19276090477691 -1.10571 -24.4697 6 17 13 0.62 0.20 - yes Open
2717 56.42485553884677 -1.20664 -21.8632 5 17 12 0.57 0.20 - yes Open
2026 56.54704593447909 -0.784632 -21.7784 9 13 0 0.00 0.00 - yes Open
2733 57.03410752473975 -1.20914 -28.1663 4 16 12 0.57 0.20 - yes Open
2725 57.766481230636224 -1.22848 -29.8795 5 17 12 0.57 0.20 - yes Open
2730 57.90645406253977 -0.982383 -22.0458 5 12 9 0.43 0.20 - yes Open
2738 59.27022752420904 -1.10992 -23.6974 8 15 9 0.43 0.20 - yes Open
2713 59.317884329959696 -1.32078 -28.2185 4 17 12 0.57 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.197kcal/mol
Ligand efficiency (LE) -0.9216kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.134
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 23HA

Physicochemical properties

Molecular weight 348.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.89
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 26.22kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 105.52kcal/mol
Minimised FF energy 79.30kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.