FAIRMol

Z56932065

Pose ID 2611 Compound 12 Pose 2611

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-1.074 kcal/mol/HA) ✓ Good fit quality (FQ -9.76) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (24.3 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-26.847
kcal/mol
LE
-1.074
kcal/mol/HA
Fit Quality
-9.76
FQ (Leeson)
HAC
25
heavy atoms
MW
376
Da
LogP
1.67
cLogP
Strain ΔE
24.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 24.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 1 Clashes 3 Severe clashes 0
Final rank3.3307698331314484Score-26.847
Inter norm-0.909233Intra norm-0.164648
Top1000noExcludedno
Contacts18H-bonds3
Artifact reasongeometry warning; 7 clashes; 3 protein contact clashes; high strain Δ 40.4
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLN36;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.86RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2619 2.425852643565488 -1.03891 -31.6075 3 17 17 0.81 0.00 - no Open
2630 2.737183101304363 -0.908696 -21.1058 1 19 19 0.90 0.00 - no Open
2610 2.87745678336561 -1.03825 -27.6698 3 16 16 0.76 0.00 - no Open
2571 3.3133375698092387 -0.781618 -18.9145 4 16 0 0.00 0.00 - no Open
2611 3.3307698331314484 -0.909233 -26.847 3 18 18 0.86 0.00 - no Current
2634 3.484222578871666 -0.90943 -19.8347 2 18 18 0.86 0.00 - no Open
2631 3.6938063235738015 -0.941899 -24.2939 2 18 18 0.86 0.00 - no Open
2579 3.842818280491077 -0.824702 -24.8535 3 16 0 0.00 0.00 - no Open
2570 4.1936771054449995 -0.920232 -24.8385 6 16 0 0.00 0.00 - no Open
2562 4.311007225668922 -0.931678 -26.7973 5 16 0 0.00 0.00 - no Open
2585 4.386769282679213 -0.924871 -23.2719 5 15 0 0.00 0.00 - no Open
2583 4.405293330625591 -0.824691 -22.8843 7 17 0 0.00 0.00 - no Open
2580 4.524655786242075 -0.883299 -21.105 5 16 0 0.00 0.00 - no Open
2561 4.755365790853137 -1.10701 -22.6931 5 18 0 0.00 0.00 - no Open
2582 5.033596954400377 -0.851607 -22.9525 4 14 0 0.00 0.00 - no Open
2574 5.14314487903842 -1.08683 -28.6837 6 14 0 0.00 0.00 - no Open
2576 5.8259569356355545 -0.916168 -25.2866 5 17 0 0.00 0.00 - no Open
2618 3.0114453068210034 -0.912672 -20.9714 2 18 18 0.86 0.00 - yes Open
2623 4.21471771581715 -0.820543 -22.0363 3 16 16 0.76 0.00 - yes Open
2639 4.248780157815152 -0.821298 -20.2188 2 16 16 0.76 0.00 - yes Open
2615 4.487514418914696 -0.882147 -25.0933 8 15 12 0.57 0.20 - yes Open
2614 4.538070645950707 -0.878637 -17.0397 2 18 18 0.86 0.00 - yes Open
2626 4.689768811513736 -0.780891 -21.8388 3 18 16 0.76 0.00 - yes Open
2635 5.067087900186418 -0.941108 -24.0972 3 18 18 0.86 0.00 - yes Open
2617 5.171769833329963 -1.09726 -25.9114 6 18 15 0.71 0.20 - yes Open
2591 5.285106474641975 -0.725459 -21.8758 1 10 0 0.00 0.00 - yes Open
2586 5.531123451872331 -1.10461 -28.6627 5 13 0 0.00 0.00 - yes Open
2564 5.6034826234630835 -0.906807 -20.5691 5 16 0 0.00 0.00 - yes Open
2577 5.787533909719497 -0.867791 -19.3597 6 18 0 0.00 0.00 - yes Open
2569 5.939339394584405 -1.05752 -26.1362 6 18 0 0.00 0.00 - yes Open
2589 5.961852564681067 -1.03278 -23.4073 7 17 0 0.00 0.00 - yes Open
2637 6.013216276604863 -1.04969 -24.6266 6 17 14 0.67 0.20 - yes Open
2590 6.246007748002172 -1.09916 -25.639 5 12 0 0.00 0.00 - yes Open
2566 6.4159852919523415 -0.92184 -23.0593 4 15 0 0.00 0.00 - yes Open
2565 6.8779477086832745 -0.861715 -8.98491 3 16 0 0.00 0.00 - yes Open
2573 7.071720201343002 -1.00754 -25.7949 6 18 0 0.00 0.00 - yes Open
2627 7.165461485168329 -0.783173 -20.7324 3 16 16 0.76 0.20 - yes Open
2563 7.321944936097866 -0.931319 -24.031 6 15 0 0.00 0.00 - yes Open
2587 7.445411535384595 -0.951119 -28.2282 6 13 0 0.00 0.00 - yes Open
2625 7.466015995483927 -1.1276 -29.6913 4 18 14 0.67 0.20 - yes Open
2620 7.548605335236438 -1.1016 -25.6395 5 19 15 0.71 0.20 - yes Open
2629 7.633404417074706 -1.15662 -26.6108 4 20 15 0.71 0.20 - yes Open
2633 7.835610140824386 -1.01254 -25.2893 4 18 15 0.71 0.20 - yes Open
2609 7.846804034211145 -1.20209 -29.4824 5 19 14 0.67 0.20 - yes Open
2572 8.011985383395809 -1.00543 -25.9321 6 17 0 0.00 0.00 - yes Open
2621 8.076562930939367 -1.07006 -25.4363 5 18 14 0.67 0.20 - yes Open
2613 8.176528115055714 -1.1272 -24.2878 4 19 14 0.67 0.20 - yes Open
2636 8.991496445453414 -1.01403 -21.282 5 18 14 0.67 0.20 - yes Open
2578 54.66175885189302 -1.16716 -32.1084 6 13 0 0.00 0.00 - yes Open
2581 54.67641370366 -1.07019 -26.8344 5 16 0 0.00 0.00 - yes Open
2616 55.79303577917653 -1.1278 -23.8755 5 19 14 0.67 0.20 - yes Open
2622 56.22232862251494 -0.826567 -18.8031 3 14 10 0.48 0.00 - yes Open
2588 56.28636613620056 -0.955578 -22.3954 7 18 0 0.00 0.00 - yes Open
2575 56.40314607127925 -0.895951 -25.702 9 13 0 0.00 0.00 - yes Open
2567 56.54258500303558 -1.02927 -28.823 6 13 0 0.00 0.00 - yes Open
2624 56.63748302183652 -0.98823 -24.9264 4 17 14 0.67 0.20 - yes Open
2568 56.75493169541731 -0.954994 -25.9646 5 18 0 0.00 0.00 - yes Open
2608 57.47118739606409 -1.05092 -28.298 4 19 15 0.71 0.20 - yes Open
2584 58.183634883560416 -0.92506 -22.6169 6 19 0 0.00 0.00 - yes Open
2638 58.259456206206714 -0.787239 -10.6807 3 15 12 0.57 0.20 - yes Open
2632 58.32206888940812 -0.928968 -20.9409 5 19 13 0.62 0.20 - yes Open
2628 58.40696538999711 -0.937958 -23.6188 4 19 14 0.67 0.20 - yes Open
2612 58.85513005734401 -1.01283 -24.2861 4 19 15 0.71 0.20 - yes Open
2560 59.13082926094182 -0.910745 -22.5104 8 20 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -26.847kcal/mol
Ligand efficiency (LE) -1.0739kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.763
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 25HA

Physicochemical properties

Molecular weight 376.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.67
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 24.28kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 100.96kcal/mol
Minimised FF energy 76.67kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.