FAIRMol

Z56781211

Pose ID 2603 Compound 254 Pose 2603

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.771 kcal/mol/HA) ✓ Good fit quality (FQ -7.36) ✗ High strain energy (14.2 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-22.369
kcal/mol
LE
-0.771
kcal/mol/HA
Fit Quality
-7.36
FQ (Leeson)
HAC
29
heavy atoms
MW
380
Da
LogP
4.32
cLogP
Strain ΔE
14.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 14.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 9 Severe clashes 0
Final rank6.19609894267377Score-22.3694
Inter norm-0.778681Intra norm0.00732317
Top1000noExcludedno
Contacts17H-bonds1
Artifact reasongeometry warning; 17 clashes; 9 protein contact clashes; high strain Δ 24.1
ResiduesA:ALA10;A:ARG29;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:THR57;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap13Native recall0.62
Jaccard0.52RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1395 4.341165307844597 -1.09547 -33.4182 9 12 0 0.00 0.00 - no Open
1389 4.698016984543662 -1.09585 -32.1976 7 13 0 0.00 0.00 - no Open
2601 5.107365695821682 -0.872555 -25.706 4 16 15 0.71 0.00 - no Open
1392 5.585988680507461 -1.08172 -29.1992 11 12 0 0.00 0.00 - no Open
1394 5.706286955061174 -1.1146 -34.3224 9 12 0 0.00 0.00 - no Open
2606 5.751229806799754 -0.984344 -27.4911 7 17 17 0.81 0.60 - no Open
2603 6.19609894267377 -0.778681 -22.3694 1 17 13 0.62 0.00 - no Current
1614 6.294594550960285 -0.802723 -25.0285 4 19 0 0.00 0.00 - no Open
1386 6.561936480504356 -1.04708 -25.0756 4 10 0 0.00 0.00 - no Open
1388 7.870389425196953 -1.06311 -27.993 5 11 0 0.00 0.00 - no Open
1610 5.523253553960511 -0.820981 -27.2929 3 20 0 0.00 0.00 - yes Open
1391 5.759179037996524 -1.15702 -34.696 9 10 0 0.00 0.00 - yes Open
1613 7.003634296654868 -0.785079 -26.2274 2 19 0 0.00 0.00 - yes Open
1611 7.368158755841646 -0.864615 -23.223 2 16 0 0.00 0.00 - yes Open
2600 7.774333813072116 -1.03515 -31.9582 4 17 17 0.81 0.40 - yes Open
2604 7.8618367838833745 -1.01334 -27.68 3 18 18 0.86 0.20 - yes Open
1387 8.298879183561594 -1.14306 -29.9025 11 14 0 0.00 0.00 - yes Open
1393 8.364608122407134 -1.19651 -31.5511 12 13 0 0.00 0.00 - yes Open
2602 8.65609965542092 -0.920343 -29.3871 3 17 17 0.81 0.20 - yes Open
1609 8.729553461477831 -0.807118 -28.8266 3 19 0 0.00 0.00 - yes Open
2607 8.763262481559165 -0.801217 -23.5699 1 13 13 0.62 0.00 - yes Open
2605 11.135925612548254 -0.862861 -24.9577 4 17 16 0.76 0.40 - yes Open
1390 12.875124913207003 -1.19523 -37.1295 4 22 0 0.00 0.00 - yes Open
1612 14.721653671734465 -0.83967 -23.0555 7 10 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.369kcal/mol
Ligand efficiency (LE) -0.7714kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.363
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 29HA

Physicochemical properties

Molecular weight 380.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.32
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 14.18kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 132.08kcal/mol
Minimised FF energy 117.90kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.