FAIRMol

Z1521553711

Pose ID 2564 Compound 24 Pose 2564

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.095 kcal/mol/HA) ✓ Good fit quality (FQ -9.34) ✓ Good H-bonds (3 bonds) ✗ High strain energy (15.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-23.005
kcal/mol
LE
-1.095
kcal/mol/HA
Fit Quality
-9.34
FQ (Leeson)
HAC
21
heavy atoms
MW
307
Da
LogP
1.71
cLogP
Strain ΔE
15.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 15.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 19 π–π 2 Clashes 9 Severe clashes 1
Final rank5.378442657506171Score-23.005
Inter norm-1.11044Intra norm0.0149684
Top1000noExcludedyes
Contacts18H-bonds3
Artifact reasonexcluded; geometry warning; 10 clashes; 1 protein clash; moderate strain Δ 15.0
ResiduesA:ALA10;A:ARG29;A:GLN36;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:THR57;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap14Native recall0.67
Jaccard0.56RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1154 1.994071832540214 -1.48556 -25.3543 7 17 0 0.00 0.00 - no Open
1152 2.432058040367128 -1.46558 -25.8481 7 17 0 0.00 0.00 - no Open
2565 2.6903141750786395 -1.17616 -22.9912 4 17 17 0.81 0.60 - no Open
1148 2.7870416321352645 -1.52737 -25.7789 7 17 0 0.00 0.00 - no Open
1150 3.1342219026699247 -1.41158 -25.2853 7 17 0 0.00 0.00 - no Open
2563 5.053100332607366 -1.05388 -22.081 3 16 12 0.57 0.00 - yes Open
2564 5.378442657506171 -1.11044 -23.005 3 18 14 0.67 0.00 - yes Current
2562 5.433527013535248 -1.09184 -21.6078 2 17 13 0.62 0.00 - yes Open
2559 6.42490854696753 -1.27478 -21.6805 3 16 13 0.62 0.20 - yes Open
2561 7.732318744832049 -1.13251 -19.9453 4 17 13 0.62 0.40 - yes Open
2566 8.330865954274609 -1.10945 -20.0265 9 19 15 0.71 0.80 - yes Open
2560 8.34233097022693 -1.1334 -20.7664 6 20 15 0.71 0.80 - yes Open
1153 8.89312562391331 -1.14068 -24.0029 5 16 0 0.00 0.00 - yes Open
1155 9.328601816548494 -1.29952 -26.6414 4 17 0 0.00 0.00 - yes Open
1151 9.735707183582283 -1.12798 -23.2641 4 17 0 0.00 0.00 - yes Open
1149 10.361254172244239 -1.2739 -25.8909 4 17 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.005kcal/mol
Ligand efficiency (LE) -1.0955kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.344
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 21HA

Physicochemical properties

Molecular weight 306.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.71
Lipinski: ≤ 5
Rotatable bonds 1

Conformational strain (MMFF94s)

Strain energy (ΔE) 15.43kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 68.09kcal/mol
Minimised FF energy 52.66kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.