FAIRMol

Z56175908

Pose ID 2555 Compound 39 Pose 2555

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.772 kcal/mol/HA) ✓ Good fit quality (FQ -7.11) ✓ Good H-bonds (4 bonds) ✗ High strain energy (18.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-20.067
kcal/mol
LE
-0.772
kcal/mol/HA
Fit Quality
-7.11
FQ (Leeson)
HAC
26
heavy atoms
MW
366
Da
LogP
5.09
cLogP
Strain ΔE
18.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 18.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 21 π–π 1 Clashes 10 Severe clashes 1
Final rank6.927600895024143Score-20.0673
Inter norm-0.865203Intra norm0.0933841
Top1000noExcludedyes
Contacts17H-bonds4
Artifact reasonexcluded; geometry warning; 13 clashes; 1 protein clash; high strain Δ 24.3
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap17Native recall0.81
Jaccard0.81RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2557 3.0053815494852105 -0.80477 -21.2544 1 18 18 0.86 0.00 - no Open
2554 3.5677614702156384 -0.94872 -24.076 2 17 17 0.81 0.40 - no Open
3372 4.365971776272748 -0.876446 -19.2495 5 14 0 0.00 0.00 - no Open
3373 4.931976348441846 -0.755071 -18.942 7 14 0 0.00 0.00 - no Open
1018 5.187462369239408 -1.2807 -32.0567 8 18 0 0.00 0.00 - no Open
1483 5.625156106846834 -1.02733 -26.3669 8 14 0 0.00 0.00 - no Open
1485 5.693204538658048 -1.04158 -26.5673 8 14 0 0.00 0.00 - no Open
1016 5.968386670347553 -1.31521 -31.1611 7 20 0 0.00 0.00 - yes Open
3371 6.131605929392736 -0.790261 -18.8721 3 14 0 0.00 0.00 - yes Open
3375 6.308087082193493 -0.79422 -20.0804 3 15 0 0.00 0.00 - yes Open
1015 6.668818675777718 -1.30204 -32.6112 4 19 0 0.00 0.00 - yes Open
3374 6.874312745205505 -0.750598 -18.3507 5 15 0 0.00 0.00 - yes Open
2555 6.927600895024143 -0.865203 -20.0673 4 17 17 0.81 0.20 - yes Current
1017 6.955192767127327 -1.31548 -33.7258 4 19 0 0.00 0.00 - yes Open
1020 7.0853352464713755 -1.17749 -28.1251 5 20 0 0.00 0.00 - yes Open
1019 7.128719430887888 -1.31509 -33.5618 3 20 0 0.00 0.00 - yes Open
1484 7.389297674496598 -0.930512 -22.3613 8 15 0 0.00 0.00 - yes Open
3376 7.702143647416033 -0.92292 -23.4018 9 14 0 0.00 0.00 - yes Open
2556 8.615207951052792 -0.907756 -23.4998 3 18 14 0.67 0.00 - yes Open
1482 9.17639228345476 -1.08029 -27.1091 9 14 0 0.00 0.00 - yes Open
1480 9.47264230357868 -1.07063 -25.3762 11 13 0 0.00 0.00 - yes Open
1481 11.93505468111776 -1.05787 -23.5819 9 18 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.067kcal/mol
Ligand efficiency (LE) -0.7718kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.111
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 365.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.09
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 18.40kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 44.70kcal/mol
Minimised FF energy 26.29kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.