FAIRMol

OHD_MAC_77

Pose ID 2451 Compound 270 Pose 2451

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.785 kcal/mol/HA) ✓ Good fit quality (FQ -7.64) ✓ Strong H-bond network (7 bonds) ✗ Very high strain energy (20.5 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-24.324
kcal/mol
LE
-0.785
kcal/mol/HA
Fit Quality
-7.64
FQ (Leeson)
HAC
31
heavy atoms
MW
419
Da
LogP
2.73
cLogP
Strain ΔE
20.5 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 20.5 kcal/mol

Interaction summary

Collapsible panels
H-bonds 7 Hydrophobic 24 π–π 4 Clashes 19 Severe clashes 5
Final rank15.730046323333022Score-24.3241
Inter norm-0.89688Intra norm0.112233
Top1000noExcludedyes
Contacts17H-bonds7
Artifact reasonexcluded; hard geometry fail; 1 severe clash; 5 protein clashes; high strain Δ 27.7
ResiduesA:ALA10;A:ARG29;A:GLU31;A:ILE139;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:THR57;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap12Native recall0.57
Jaccard0.46RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role2Role recall0.40
H-bond same residue2Residue recall0.40

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2456 5.249819782812001 -0.74814 -20.1545 3 19 17 0.81 0.40 - no Open
1751 6.387594634546211 -0.675974 -17.3507 5 16 0 0.00 0.00 - no Open
2457 6.407277374141122 -0.74922 -20.2182 7 17 14 0.67 0.20 - no Open
1785 6.449351689377192 -0.510179 -10.5795 5 10 0 0.00 0.00 - no Open
1783 6.638877622320285 -0.619022 -11.522 7 11 0 0.00 0.00 - no Open
2454 7.379286366834068 -0.852848 -17.5947 7 18 16 0.76 0.20 - no Open
3160 8.767937290115395 -0.697321 -12.7011 6 15 0 0.00 0.00 - no Open
1284 9.85179150053064 -0.983283 -23.5196 16 22 0 0.00 0.00 - no Open
1784 7.322761670305217 -0.577814 -18.0294 4 13 0 0.00 0.00 - yes Open
3163 7.822885735839338 -0.73556 -17.8161 4 15 0 0.00 0.00 - yes Open
1786 7.8404161504482355 -0.489006 -13.7238 7 7 0 0.00 0.00 - yes Open
2455 7.9521670430524845 -0.788095 -15.5652 4 17 15 0.71 0.20 - yes Open
1749 8.286378000269185 -0.591758 -9.93257 6 14 0 0.00 0.00 - yes Open
1747 8.359125435996447 -0.741136 -13.7987 7 14 0 0.00 0.00 - yes Open
3159 8.411444974025983 -0.773706 -22.989 7 17 0 0.00 0.00 - yes Open
3158 8.536688175904015 -0.730265 -15.9603 7 13 0 0.00 0.00 - yes Open
3161 8.637492496517854 -0.72337 -15.6539 10 17 0 0.00 0.00 - yes Open
1752 8.900089661808044 -0.833214 -13.3981 7 14 0 0.00 0.00 - yes Open
1280 8.997939519386627 -1.00788 -22.242 13 20 0 0.00 0.00 - yes Open
1787 9.03616053002429 -0.590656 -14.175 8 11 0 0.00 0.00 - yes Open
1748 9.265549701808197 -0.689773 -17.7272 12 13 0 0.00 0.00 - yes Open
1281 9.399523811169527 -0.947312 -17.127 13 22 0 0.00 0.00 - yes Open
2452 9.749041312581422 -0.774831 -20.9279 4 17 14 0.67 0.00 - yes Open
1278 9.782975491762757 -1.01011 -29.4453 16 24 0 0.00 0.00 - yes Open
1782 9.902278180314955 -0.802503 -18.6827 9 14 0 0.00 0.00 - yes Open
1750 10.113433440849207 -0.515959 -11.9296 8 14 0 0.00 0.00 - yes Open
3162 10.46717236152207 -0.599199 -14.3565 4 16 0 0.00 0.00 - yes Open
2453 11.406159126158812 -0.747023 -13.5772 5 18 16 0.76 0.20 - yes Open
1277 12.347568068203564 -0.933548 -20.8237 16 23 0 0.00 0.00 - yes Open
1283 12.715725545062385 -0.980705 -23.9407 16 23 0 0.00 0.00 - yes Open
1279 12.868678692629699 -0.786475 -17.5772 15 22 0 0.00 0.00 - yes Open
3164 13.066728051042078 -0.731 -14.6911 5 17 0 0.00 0.00 - yes Open
1282 13.669630427519559 -0.861208 -20.8788 16 21 0 0.00 0.00 - yes Open
2451 15.730046323333022 -0.89688 -24.3241 7 17 12 0.57 0.40 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.324kcal/mol
Ligand efficiency (LE) -0.7846kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.644
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 31HA

Physicochemical properties

Molecular weight 419.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.73
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 20.48kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 89.57kcal/mol
Minimised FF energy 69.09kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.