FAIRMol

OHD_MAC_26

Pose ID 2308 Compound 335 Pose 2308

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.654 kcal/mol/HA) ✓ Good fit quality (FQ -6.64) ✗ Very high strain energy (36.6 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-23.535
kcal/mol
LE
-0.654
kcal/mol/HA
Fit Quality
-6.64
FQ (Leeson)
HAC
36
heavy atoms
MW
521
Da
LogP
4.69
cLogP
Strain ΔE
36.6 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 36.6 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 3 Clashes 8 Severe clashes 0
Final rank6.626389575561139Score-23.5345
Inter norm-0.764599Intra norm0.110863
Top1000noExcludedno
Contacts17H-bonds2
Artifact reasongeometry warning; 16 clashes; 8 protein contact clashes; high strain Δ 40.5
ResiduesA:ARG29;A:ASN65;A:GLN36;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR57;A:VAL116

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap14Native recall0.67
Jaccard0.58RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2310 5.825908708628535 -0.64971 -18.6671 0 21 17 0.81 0.00 - no Open
2308 6.626389575561139 -0.764599 -23.5345 2 17 14 0.67 0.20 - no Current
3152 6.870321733375402 -0.557739 -19.7623 4 15 0 0.00 0.00 - no Open
1319 8.116023195184516 -0.600381 -17.4612 2 12 0 0.00 0.00 - no Open
1112 8.958969797044404 -0.679215 -21.5065 10 19 0 0.00 0.00 - no Open
1111 9.154012993422636 -0.790874 -21.8518 9 23 0 0.00 0.00 - no Open
1320 7.144697201093516 -0.66438 -23.2682 4 17 0 0.00 0.00 - yes Open
2311 10.696089840028915 -0.783533 -24.9492 5 19 15 0.71 0.20 - yes Open
3154 11.19188595623392 -0.601709 -14.8051 3 15 0 0.00 0.00 - yes Open
2309 11.436404437618762 -0.827759 -21.9922 5 21 16 0.76 0.40 - yes Open
3153 12.604935622414184 -0.482364 -5.50888 4 15 0 0.00 0.00 - yes Open
3155 13.136139902746507 -0.680116 -24.0446 4 19 0 0.00 0.00 - yes Open
1110 13.494986240004152 -0.778033 -22.8904 12 21 0 0.00 0.00 - yes Open
1113 13.996316682324466 -0.935175 -30.3559 12 21 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.535kcal/mol
Ligand efficiency (LE) -0.6537kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.644
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 36HA

Physicochemical properties

Molecular weight 521.0Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.69
Lipinski: ≤ 5
Rotatable bonds 9

Conformational strain (MMFF94s)

Strain energy (ΔE) 36.57kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 155.69kcal/mol
Minimised FF energy 119.12kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.