FAIRMol

Z44831334

Pose ID 20090 Compound 1669 Pose 2284

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.675 kcal/mol/HA) ✓ Good fit quality (FQ -6.37) ✓ Strong H-bond network (8 bonds) ✗ High strain energy (17.9 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-18.901
kcal/mol
LE
-0.675
kcal/mol/HA
Fit Quality
-6.37
FQ (Leeson)
HAC
28
heavy atoms
MW
374
Da
LogP
3.31
cLogP
Strain ΔE
17.9 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 8 Hydrophobic 11 π–π 3 Clashes 6 Severe clashes 0
Final rank4.3247306630238604Score-18.9013
Inter norm-0.692287Intra norm0.0172413
Top1000noExcludedno
Contacts21H-bonds8
Artifact reasongeometry warning; 13 clashes; 6 protein contact clashes; moderate strain Δ 18.7
ResiduesA:ALA15;A:ARG116;A:ARG140;A:ARG144;A:ASN106;A:ASP13;A:CYS72;A:GLN100;A:GLN104;A:GLY73;A:GLY75;A:GLY77;A:HIS105;A:HIS14;A:HIS141;A:ILE76;A:LEU101;A:LEU136;A:THR74;A:TYR49;A:VAL97

Protein summary

155 residues
Protein targetT10Atoms4590
Residues155Chains1
Residue summaryILE:494; ARG:384; ALA:360; VAL:352; LEU:304; GLU:300; THR:280; MET:272; LYS:220; ASP:216; TYR:210; HIS:204; GLY:182; SER:176; GLN:170; ASN:140

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6FXWContacts17
PoseOpen native poseH-bonds16
IFP residuesA:ALA15; A:ARG116; A:ARG140; A:ARG144; A:ASN106; A:ASP13; A:CYS72; A:GLY73; A:GLY75; A:GLY77; A:HIS105; A:HIS14; A:HIS141; A:ILE76; A:LEU101; A:THR74; A:TYR49
Current overlap17Native recall1.00
Jaccard0.81RMSD-
H-bond strict4Strict recall0.31
H-bond same residue+role6Role recall0.55
H-bond same residue6Residue recall0.55

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2284 4.3247306630238604 -0.692287 -18.9013 8 21 17 1.00 0.55 - no Current
2292 4.360250085050621 -0.768671 -19.1246 7 19 17 1.00 0.36 - no Open
2282 4.7249650172378885 -0.729074 -11.1741 4 15 12 0.71 0.27 - no Open
1966 4.747523612073444 -1.04185 -23.4341 10 16 0 0.00 0.00 - no Open
1956 5.32512624871409 -1.06121 -20.2321 5 16 0 0.00 0.00 - no Open
2283 5.632559324072815 -0.888374 -21.6551 10 18 15 0.88 0.36 - no Open
1777 6.1830308088073656 -1.02278 -28.9521 6 11 0 0.00 0.00 - no Open
2288 6.375013859983085 -0.70968 -20.857 8 21 17 1.00 0.45 - no Open
2298 6.7145536812605515 -0.80443 -17.7347 8 18 15 0.88 0.36 - no Open
1959 6.935256137375159 -1.01124 -21.3057 10 11 0 0.00 0.00 - no Open
1770 5.094517942437423 -0.776275 -21.5357 6 17 0 0.00 0.00 - yes Open
1781 5.993714358976294 -0.963848 -25.2427 7 10 0 0.00 0.00 - yes Open
2293 6.2440871409905165 -0.933802 -18.8054 13 17 16 0.94 0.45 - yes Open
1968 6.5192963449486125 -1.07734 -29.3409 4 17 0 0.00 0.00 - yes Open
2296 6.670196227444615 -0.65908 -18.8552 6 19 15 0.88 0.36 - yes Open
1769 6.678946686528415 -1.15568 -31.5114 5 20 0 0.00 0.00 - yes Open
2285 7.149219817082675 -1.07304 -31.4732 8 15 14 0.82 0.45 - yes Open
1972 7.181469421543011 -1.14544 -32.154 8 16 0 0.00 0.00 - yes Open
1973 7.288714480071388 -1.05791 -27.3986 6 17 0 0.00 0.00 - yes Open
2294 7.326789476286028 -0.65423 -13.8044 6 16 13 0.76 0.27 - yes Open
1767 7.521536317925812 -1.03902 -25.424 6 22 0 0.00 0.00 - yes Open
2299 7.540412476316772 -0.978304 -22.2374 11 15 15 0.88 0.45 - yes Open
1955 7.54817879027187 -1.11572 -26.3431 7 17 0 0.00 0.00 - yes Open
1765 7.578259528912266 -1.11777 -29.6718 11 15 0 0.00 0.00 - yes Open
2287 7.615465620804151 -1.10593 -34.1592 9 14 14 0.82 0.45 - yes Open
1779 7.932511813137621 -1.03276 -23.3051 5 20 0 0.00 0.00 - yes Open
1772 8.03479195823699 -1.10109 -23.508 6 18 0 0.00 0.00 - yes Open
1764 8.285695152840127 -1.06504 -19.0839 5 17 0 0.00 0.00 - yes Open
1780 8.35350700049101 -1.0302 -22.9431 7 20 0 0.00 0.00 - yes Open
1974 8.582276928256347 -1.19801 -29.6594 4 19 0 0.00 0.00 - yes Open
1768 8.853169226990572 -1.20186 -32.6137 5 20 0 0.00 0.00 - yes Open
2290 8.957338923391148 -0.728737 -7.8102 5 17 12 0.71 0.18 - yes Open
2300 8.986220175570722 -0.877553 -21.7457 10 13 11 0.65 0.36 - yes Open
1773 9.263326875679725 -0.979622 -25.6234 6 14 0 0.00 0.00 - yes Open
2289 9.356842411316178 -0.765645 -12.7259 12 15 11 0.65 0.36 - yes Open
1965 9.495910905989886 -1.13479 -28.3845 8 11 0 0.00 0.00 - yes Open
1776 9.543027710748651 -1.03583 -18.8836 6 20 0 0.00 0.00 - yes Open
1960 9.891393855116439 -1.18648 -30.2597 11 20 0 0.00 0.00 - yes Open
1762 10.030869945109714 -0.809182 -15.4188 7 17 0 0.00 0.00 - yes Open
1967 10.423596973533662 -0.96711 -18.1403 7 17 0 0.00 0.00 - yes Open
1775 10.691282540875303 -1.06431 -30.9539 6 13 0 0.00 0.00 - yes Open
1964 11.72168746396509 -1.12267 -23.1435 10 20 0 0.00 0.00 - yes Open
1961 12.298260188871199 -1.04957 -29.7574 4 18 0 0.00 0.00 - yes Open
1958 12.435688708889908 -1.22174 -31.2061 8 18 0 0.00 0.00 - yes Open
1969 13.695405501477392 -1.09595 -24.824 5 22 0 0.00 0.00 - yes Open
2281 57.390183518013785 -0.966606 -21.753 12 16 16 0.94 0.45 - yes Open
2295 57.9014749728669 -0.943467 -23.6847 11 16 14 0.82 0.45 - yes Open
1971 58.09867251574792 -1.04126 -23.6899 8 17 0 0.00 0.00 - yes Open
2291 58.36702646729543 -0.837258 -19.9376 10 13 12 0.71 0.55 - yes Open
2286 58.43071512599702 -0.882818 -22.4478 9 17 17 1.00 0.36 - yes Open
1778 58.791991872409916 -0.966466 -17.1018 7 20 0 0.00 0.00 - yes Open
2297 59.01480915496941 -0.973727 -22.5506 11 15 15 0.88 0.45 - yes Open
1771 59.84187762441071 -1.04123 -30.7734 6 13 0 0.00 0.00 - yes Open
1766 60.631817711192944 -0.91319 -24.2612 7 20 0 0.00 0.00 - yes Open
1763 60.653579440356104 -1.07234 -31.3119 6 13 0 0.00 0.00 - yes Open
1774 60.92032805873688 -0.771161 -11.7976 6 20 0 0.00 0.00 - yes Open
1962 62.117610681833504 -1.08667 -30.5238 8 18 0 0.00 0.00 - yes Open
1957 63.51845393719181 -1.07379 -22.2037 9 21 0 0.00 0.00 - yes Open
1970 63.52779421384398 -1.26163 -35.075 9 17 0 0.00 0.00 - yes Open
1963 64.85238330100844 -0.954113 -12.9002 8 19 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -18.901kcal/mol
Ligand efficiency (LE) -0.6750kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.373
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 28HA

Physicochemical properties

Molecular weight 374.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.31
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 17.88kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 111.60kcal/mol
Minimised FF energy 93.72kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.