FAIRMol

TC488

Pose ID 1994 Compound 404 Pose 1994

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.624 kcal/mol/HA) ✓ Good fit quality (FQ -6.44) ✓ Good H-bonds (3 bonds) ✗ High strain energy (18.3 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-23.723
kcal/mol
LE
-0.624
kcal/mol/HA
Fit Quality
-6.44
FQ (Leeson)
HAC
38
heavy atoms
MW
516
Da
LogP
3.89
cLogP
Strain ΔE
18.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 18.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 3 Clashes 7 Severe clashes 2
Final rank57.51677514441389Score-23.7228
Inter norm-0.583446Intra norm-0.0408382
Top1000noExcludedyes
Contacts17H-bonds3
Artifact reasonexcluded; geometry warning; 17 clashes; 2 protein clashes
ResiduesA:ALA10;A:ASN65;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap15Native recall0.71
Jaccard0.65RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1224 4.655005214225548 -0.484602 -15.5856 2 11 0 0.00 0.00 - no Open
1014 5.105019058142142 -0.605348 -19.8969 6 18 0 0.00 0.00 - no Open
1221 6.370386724896184 -0.41635 -15.1312 5 14 0 0.00 0.00 - no Open
669 6.400172688267178 -0.762569 -25.878 8 15 0 0.00 0.00 - no Open
1991 7.051437491616422 -0.681096 -25.1495 5 18 14 0.67 0.00 - no Open
1222 6.531760830123513 -0.573627 -18.5949 2 15 0 0.00 0.00 - yes Open
1993 7.119321826583064 -0.687894 -19.7625 3 18 16 0.76 0.00 - yes Open
1011 7.659122942096789 -0.624349 -21.4721 3 21 0 0.00 0.00 - yes Open
1016 7.715255248601405 -0.599842 -24.1332 5 15 0 0.00 0.00 - yes Open
1992 8.065732105702462 -0.571842 -23.1664 5 19 15 0.71 0.40 - yes Open
667 8.536720782848368 -0.821892 -27.8573 6 15 0 0.00 0.00 - yes Open
1223 8.630879763671473 -0.499288 -19.2264 3 14 0 0.00 0.00 - yes Open
1012 9.126618597058714 -0.669323 -26.5351 2 19 0 0.00 0.00 - yes Open
670 9.52214347548418 -0.829467 -25.5867 7 17 0 0.00 0.00 - yes Open
671 10.207353193760811 -0.787479 -27.9037 0 21 0 0.00 0.00 - yes Open
1015 10.554637340146453 -0.765696 -21.0966 8 15 0 0.00 0.00 - yes Open
1225 10.660258035923938 -0.601518 -17.8603 5 15 0 0.00 0.00 - yes Open
666 13.90791226219642 -0.782514 -24.566 7 16 0 0.00 0.00 - yes Open
1994 57.51677514441389 -0.583446 -23.7228 3 17 15 0.71 0.00 - yes Current
1226 58.23524297792672 -0.569285 -21.0713 4 16 0 0.00 0.00 - yes Open
1013 59.332862727416845 -0.566977 -18.5546 6 15 0 0.00 0.00 - yes Open
668 63.28941991823524 -0.744512 -20.497 7 16 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.723kcal/mol
Ligand efficiency (LE) -0.6243kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.436
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 38HA

Physicochemical properties

Molecular weight 515.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.89
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 18.33kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 94.51kcal/mol
Minimised FF energy 76.18kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.