FAIRMol

Z46032342

Pose ID 19800 Compound 2015 Pose 1994

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.580 kcal/mol/HA) ✓ Good fit quality (FQ -4.95) ✓ Good H-bonds (3 bonds) ✗ High strain energy (11.7 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-12.182
kcal/mol
LE
-0.580
kcal/mol/HA
Fit Quality
-4.95
FQ (Leeson)
HAC
21
heavy atoms
MW
282
Da
LogP
3.06
cLogP
Strain ΔE
11.7 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 4 π–π 1 Clashes 6 Severe clashes 0 ⚠ Hydrophobic exposure 52%
⚠️Partial hydrophobic solvent exposure
53% of hydrophobic surface appears solvent-exposed (9/17 atoms). Partial exposure is common but may limit selectivity and membrane permeability.
Non-polar atoms 17 Buried (contacted) 8 Exposed 9 LogP 3.06 H-bonds 3
Exposed fragments: phenyl (6/6 atoms exposed)aliphatic chain/group (3 atoms exposed)
Final rank3.4010284562600055Score-12.1824
Inter norm-0.789216Intra norm0.2091
Top1000noExcludedno
Contacts14H-bonds3
Artifact reasongeometry warning; 10 clashes; 6 protein contact clashes
ResiduesA:ALA15;A:ARG116;A:ARG140;A:ARG144;A:ASN106;A:ASP13;A:CYS72;A:GLY73;A:HIS105;A:HIS14;A:HIS141;A:SER46;A:THR74;A:TYR49

Protein summary

155 residues
Protein targetT10Atoms4590
Residues155Chains1
Residue summaryILE:494; ARG:384; ALA:360; VAL:352; LEU:304; GLU:300; THR:280; MET:272; LYS:220; ASP:216; TYR:210; HIS:204; GLY:182; SER:176; GLN:170; ASN:140

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6FXWContacts17
PoseOpen native poseH-bonds16
IFP residuesA:ALA15; A:ARG116; A:ARG140; A:ARG144; A:ASN106; A:ASP13; A:CYS72; A:GLY73; A:GLY75; A:GLY77; A:HIS105; A:HIS14; A:HIS141; A:ILE76; A:LEU101; A:THR74; A:TYR49
Current overlap13Native recall0.76
Jaccard0.72RMSD-
H-bond strict2Strict recall0.15
H-bond same residue+role2Role recall0.18
H-bond same residue3Residue recall0.27

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1994 3.4010284562600055 -0.789216 -12.1824 3 14 13 0.76 0.18 - no Current
1993 5.581058656508104 -1.09845 -18.5398 6 15 15 0.88 0.27 - yes Open
1992 5.774768438519566 -1.00354 -13.8413 9 17 16 0.94 0.36 - yes Open
1995 11.036989953241015 -0.914927 -17.9317 5 15 15 0.88 0.36 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -12.182kcal/mol
Ligand efficiency (LE) -0.5801kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.948
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 21HA

Physicochemical properties

Molecular weight 282.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.06
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 11.69kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 83.00kcal/mol
Minimised FF energy 71.31kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.