FAIRMol

Z46589685

Pose ID 19465 Compound 793 Pose 1659

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.821 kcal/mol/HA) ✓ Good fit quality (FQ -7.75) ✓ Strong H-bond network (6 bonds) ✗ High strain energy (17.6 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-22.988
kcal/mol
LE
-0.821
kcal/mol/HA
Fit Quality
-7.75
FQ (Leeson)
HAC
28
heavy atoms
MW
401
Da
LogP
3.56
cLogP
Strain ΔE
17.6 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 6 Hydrophobic 6 π–π 3 Clashes 4 Severe clashes 0 ⚠ Hydrophobic exposure 42%
⚠️Partial hydrophobic solvent exposure
43% of hydrophobic surface appears solvent-exposed (9/21 atoms). Partial exposure is common but may limit selectivity and membrane permeability.
Non-polar atoms 21 Buried (contacted) 12 Exposed 9 LogP 3.56 H-bonds 6
Exposed fragments: phenyl (6/7 atoms exposed)aliphatic chain/group (3 atoms exposed)
Final rank3.56564033182907Score-22.9885
Inter norm-0.782688Intra norm-0.0383288
Top1000noExcludedno
Contacts17H-bonds6
Artifact reasongeometry warning; 9 clashes; 4 protein contact clashes; high strain Δ 27.2
ResiduesA:ALA15;A:ARG116;A:ARG140;A:ARG144;A:ASN106;A:ASP13;A:CYS72;A:GLY73;A:GLY75;A:GLY77;A:HIS105;A:HIS14;A:HIS141;A:ILE76;A:LEU101;A:THR74;A:TYR49

Protein summary

155 residues
Protein targetT10Atoms4590
Residues155Chains1
Residue summaryILE:494; ARG:384; ALA:360; VAL:352; LEU:304; GLU:300; THR:280; MET:272; LYS:220; ASP:216; TYR:210; HIS:204; GLY:182; SER:176; GLN:170; ASN:140

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6FXWContacts17
PoseOpen native poseH-bonds16
IFP residuesA:ALA15; A:ARG116; A:ARG140; A:ARG144; A:ASN106; A:ASP13; A:CYS72; A:GLY73; A:GLY75; A:GLY77; A:HIS105; A:HIS14; A:HIS141; A:ILE76; A:LEU101; A:THR74; A:TYR49
Current overlap17Native recall1.00
Jaccard1.00RMSD-
H-bond strict3Strict recall0.23
H-bond same residue+role3Role recall0.27
H-bond same residue5Residue recall0.45

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1134 2.216689295671921 -0.834277 -22.7818 3 11 0 0.00 0.00 - no Open
1663 3.2881602176397022 -0.677526 -18.9897 7 17 17 1.00 0.27 - no Open
1659 3.56564033182907 -0.782688 -22.9885 6 17 17 1.00 0.27 - no Current
1136 5.32045043821675 -0.794006 -13.9832 8 13 0 0.00 0.00 - no Open
1660 6.053762675317191 -0.665169 -14.3171 4 17 15 0.88 0.09 - no Open
1135 4.31633562251834 -0.817233 -20.0377 6 13 0 0.00 0.00 - yes Open
1133 5.968579536806257 -0.850383 -19.6588 5 12 0 0.00 0.00 - yes Open
1661 6.811133083225781 -0.621708 -16.2631 7 14 13 0.76 0.36 - yes Open
1138 6.8125916135845594 -0.838168 -23.0405 6 12 0 0.00 0.00 - yes Open
1662 7.6094390736925845 -0.724771 -15.4222 7 17 16 0.94 0.36 - yes Open
1137 9.291740465870225 -0.709112 -17.2553 6 13 0 0.00 0.00 - yes Open
1658 11.337302085200848 -0.768955 -16.9716 8 15 14 0.82 0.45 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.988kcal/mol
Ligand efficiency (LE) -0.8210kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.751
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 28HA

Physicochemical properties

Molecular weight 401.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.56
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 17.62kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 5.27kcal/mol
Minimised FF energy -12.35kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.