FAIRMol

TC228

Pose ID 1944 Compound 401 Pose 1944

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good LE (-0.328 kcal/mol/HA) ✓ Good fit quality (FQ -3.59) ✓ Strong H-bond network (6 bonds) ✗ Very high strain energy (51.6 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-16.075
kcal/mol
LE
-0.328
kcal/mol/HA
Fit Quality
-3.59
FQ (Leeson)
HAC
49
heavy atoms
MW
696
Da
LogP
4.28
cLogP
Strain ΔE
51.6 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: good
Geometry reliability: low
Reason: geometry warning, clashes, strain 51.6 kcal/mol

Interaction summary

Collapsible panels
H-bonds 6 Hydrophobic 24 π–π 0 Clashes 6 Severe clashes 2
Final rank8.662739610179079Score-16.0745
Inter norm-0.408119Intra norm0.0800681
Top1000noExcludedyes
Contacts22H-bonds6
Artifact reasonexcluded; geometry warning; 9 clashes; 2 protein clashes; high strain Δ 52.3
ResiduesA:ALA10;A:ARG29;A:ASN65;A:ASP22;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:LYS64;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap17Native recall0.81
Jaccard0.65RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1942 7.036449674784217 -0.447771 -16.702 4 20 16 0.76 0.20 - no Open
1944 8.662739610179079 -0.408119 -16.0745 6 22 17 0.81 0.00 - yes Current
1943 10.890201577728417 -0.430146 -20.3116 2 20 18 0.86 0.20 - yes Open
1941 58.869974284176465 -0.586001 -25.7654 7 20 17 0.81 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -16.075kcal/mol
Ligand efficiency (LE) -0.3281kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -3.590
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 49HA

Physicochemical properties

Molecular weight 695.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.28
Lipinski: ≤ 5
Rotatable bonds 13

Conformational strain (MMFF94s)

Strain energy (ΔE) 51.56kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 110.31kcal/mol
Minimised FF energy 58.76kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.