FAIRMol

ulfkktlib_3721

Pose ID 1888 Compound 341 Pose 1888

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.668 kcal/mol/HA) ✓ Good fit quality (FQ -6.68) ✗ Very high strain energy (90.2 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-22.706
kcal/mol
LE
-0.668
kcal/mol/HA
Fit Quality
-6.68
FQ (Leeson)
HAC
34
heavy atoms
MW
458
Da
LogP
2.03
cLogP
Strain ΔE
90.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 90.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 9 Severe clashes 1
Final rank54.820022768434065Score-22.7058
Inter norm-0.715126Intra norm0.0473098
Top1000noExcludedyes
Contacts19H-bonds1
Artifact reasonexcluded; geometry warning; 6 clashes; 1 protein clash
ResiduesA:ALA10;A:ASN65;A:GLN36;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO62;A:SER60;A:THR137;A:THR57;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.82RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1889 5.941232072190054 -0.653889 -16.9133 1 18 14 0.67 0.20 - no Open
1893 6.293968436080832 -0.665763 -21.2699 1 18 15 0.71 0.20 - no Open
755 6.4389098311611 -0.910539 -23.9467 2 14 0 0.00 0.00 - no Open
1892 7.037379092237105 -0.758403 -25.9095 1 19 15 0.71 0.00 - no Open
756 9.304039898740802 -0.897508 -26.7825 4 13 0 0.00 0.00 - no Open
754 9.582377568419362 -0.83118 -24.4702 2 15 0 0.00 0.00 - yes Open
1888 54.820022768434065 -0.715126 -22.7058 1 19 18 0.86 0.20 - yes Current
757 55.0167620659418 -0.793948 -25.8005 2 14 0 0.00 0.00 - yes Open
1891 55.07199189602411 -0.715341 -22.2772 2 19 15 0.71 0.20 - yes Open
758 55.11195747090152 -0.8265 -27.3864 3 18 0 0.00 0.00 - yes Open
759 56.5538067791244 -0.910616 -25.7559 3 15 0 0.00 0.00 - yes Open
1890 58.59615633900195 -0.66757 -19.8007 4 20 17 0.81 0.40 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.706kcal/mol
Ligand efficiency (LE) -0.6678kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.682
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 457.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.03
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 90.23kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 284.90kcal/mol
Minimised FF energy 194.67kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.