FAIRMol

OHD_Leishmania_259

Pose ID 17825 Compound 2013 Pose 19

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.097 kcal/mol/HA) ✓ Good fit quality (FQ -9.36) ✓ Strong H-bond network (9 bonds) ✗ High strain energy (16.4 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-23.035
kcal/mol
LE
-1.097
kcal/mol/HA
Fit Quality
-9.36
FQ (Leeson)
HAC
21
heavy atoms
MW
286
Da
LogP
3.07
cLogP
Strain ΔE
16.4 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 9 Hydrophobic 5 π–π 1 Clashes 7 Severe clashes 0 ⚠ Hydrophobic exposure 60%
🚨Solvent-exposed hydrophobic surface — desolvation penalty likely
60% of hydrophobic surface is solvent-exposed (9/15 atoms). Large non-polar area without protein contacts incurs a desolvation penalty and will reduce binding affinity. Consider truncating or replacing the exposed fragment.
Non-polar atoms 15 Buried (contacted) 6 Exposed 9 LogP 3.07 H-bonds 9
Exposed fragments: phenyl (6/6 atoms exposed)aliphatic chain/group (3 atoms exposed)
Final rank3.1437733935534817Score-23.0349
Inter norm-1.25666Intra norm0.159758
Top1000noExcludedno
Contacts16H-bonds9
Artifact reasongeometry warning; 8 clashes; 7 protein contact clashes; moderate strain Δ 17.5
ResiduesA:ALA15;A:ARG116;A:ARG140;A:ARG144;A:ASN106;A:ASP13;A:CYS72;A:GLY73;A:GLY75;A:GLY77;A:HIS105;A:HIS14;A:HIS141;A:ILE76;A:THR74;A:TYR49

Protein summary

155 residues
Protein targetT10Atoms4590
Residues155Chains1
Residue summaryILE:494; ARG:384; ALA:360; VAL:352; LEU:304; GLU:300; THR:280; MET:272; LYS:220; ASP:216; TYR:210; HIS:204; GLY:182; SER:176; GLN:170; ASN:140

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6FXWContacts17
PoseOpen native poseH-bonds16
IFP residuesA:ALA15; A:ARG116; A:ARG140; A:ARG144; A:ASN106; A:ASP13; A:CYS72; A:GLY73; A:GLY75; A:GLY77; A:HIS105; A:HIS14; A:HIS141; A:ILE76; A:LEU101; A:THR74; A:TYR49
Current overlap16Native recall0.94
Jaccard0.94RMSD-
H-bond strict5Strict recall0.38
H-bond same residue+role4Role recall0.36
H-bond same residue6Residue recall0.55

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
58 2.7306715585041426 -1.06088 -20.3608 7 14 0 0.00 0.00 - no Open
19 3.1437733935534817 -1.25666 -23.0349 9 16 16 0.94 0.36 - no Current
56 4.458122118916195 -1.12271 -21.4642 12 16 1 0.06 0.00 - no Open
20 5.161952373505933 -0.974176 -18.0396 9 14 13 0.76 0.45 - no Open
57 5.12760702112999 -0.946948 -17.8172 10 16 0 0.00 0.00 - yes Open
21 5.5231088854595445 -1.25733 -21.3816 9 16 16 0.94 0.36 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.035kcal/mol
Ligand efficiency (LE) -1.0969kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.356
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 21HA

Physicochemical properties

Molecular weight 286.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.07
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 16.36kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 78.33kcal/mol
Minimised FF energy 61.96kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.