FAIRMol

OSA_Lib_303

Pose ID 1771 Compound 76 Pose 1771

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.808 kcal/mol/HA) ✓ Good fit quality (FQ -7.80) ✗ Very high strain energy (22.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-24.247
kcal/mol
LE
-0.808
kcal/mol/HA
Fit Quality
-7.80
FQ (Leeson)
HAC
30
heavy atoms
MW
399
Da
LogP
3.81
cLogP
Strain ΔE
22.4 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 3 Clashes 9 Severe clashes 2
Final rank57.31615126997281Score-24.247
Inter norm-0.932011Intra norm0.123776
Top1000noExcludedyes
Contacts18H-bonds2
Artifact reasonexcluded; geometry warning; 15 clashes; 2 protein clashes
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO62;A:SER60;A:THR57;A:TRP25;A:TYR122;A:VAL116

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap16Native recall0.76
Jaccard0.70RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1774 3.573288050063608 -0.772999 -21.9004 2 20 17 0.81 0.00 - no Open
2504 3.660721520100676 -0.729517 -21.5858 1 17 0 0.00 0.00 - no Open
1862 3.87219139404224 -0.815061 -23.24 1 17 0 0.00 0.00 - no Open
1859 4.044797902455198 -0.841637 -24.6125 2 16 0 0.00 0.00 - no Open
1775 4.083144695775258 -0.728624 -21.6912 1 16 14 0.67 0.00 - no Open
1853 4.10184010020892 -0.880758 -27.1162 2 20 0 0.00 0.00 - no Open
1867 4.119210628346155 -0.827872 -25.7791 2 19 0 0.00 0.00 - no Open
2510 4.1921996790157605 -0.70955 -21.5318 1 16 0 0.00 0.00 - no Open
666 4.2026533814878615 -1.07778 -24.1679 3 17 0 0.00 0.00 - no Open
1769 4.306591512368701 -0.764589 -21.6771 1 17 14 0.67 0.00 - no Open
1856 4.44984162506596 -0.826813 -25.0381 2 19 0 0.00 0.00 - no Open
1865 4.489069700446324 -0.853108 -26.2028 2 16 0 0.00 0.00 - no Open
1857 4.60207313262103 -0.870965 -25.5233 2 19 0 0.00 0.00 - no Open
1860 4.941176211073369 -0.814242 -23.1829 1 19 0 0.00 0.00 - no Open
2512 4.9499879180043935 -0.533637 -15.8118 1 14 0 0.00 0.00 - no Open
1772 5.084244868679373 -0.720538 -19.5788 1 17 14 0.67 0.00 - no Open
2515 5.08998407023543 -0.723521 -21.8715 2 17 0 0.00 0.00 - no Open
1770 5.539903271014922 -0.661452 -20.0834 1 17 15 0.71 0.20 - no Open
672 5.609142162413652 -0.97887 -28.4095 0 18 0 0.00 0.00 - no Open
1777 5.827949941320511 -0.826804 -24.4048 1 20 19 0.90 0.20 - no Open
2507 6.028855781518878 -0.674504 -18.8887 2 13 0 0.00 0.00 - no Open
670 6.069152296260166 -0.848161 -20.0064 2 20 0 0.00 0.00 - no Open
1861 54.23584161740301 -0.866582 -27.591 2 19 0 0.00 0.00 - no Open
671 55.84034710540824 -1.0461 -31.3666 3 16 0 0.00 0.00 - no Open
2513 56.752684427219364 -0.511399 -15.524 1 12 0 0.00 0.00 - no Open
669 57.88244178748334 -0.876207 -24.1328 3 16 0 0.00 0.00 - no Open
1855 7.426943019173197 -0.821617 -22.7875 1 15 0 0.00 0.00 - yes Open
2505 7.663017115939302 -0.746292 -21.2169 4 13 0 0.00 0.00 - yes Open
1868 53.97468230510326 -0.855091 -27.5803 1 14 0 0.00 0.00 - yes Open
1866 55.06104951731334 -0.84078 -25.006 1 16 0 0.00 0.00 - yes Open
2509 55.63878368400333 -0.708493 -20.9189 1 17 0 0.00 0.00 - yes Open
2508 55.73331777063794 -0.650146 -18.1186 4 13 0 0.00 0.00 - yes Open
1780 55.80983335278023 -0.740289 -22.3618 0 20 19 0.90 0.00 - yes Open
1779 55.99983980577713 -0.680155 -19.0918 1 17 14 0.67 0.00 - yes Open
2514 56.14429881458122 -0.634465 -17.5186 2 12 0 0.00 0.00 - yes Open
665 56.26304349817779 -0.970114 -28.504 1 18 0 0.00 0.00 - yes Open
668 56.38329802096 -0.64718 -18.107 1 11 0 0.00 0.00 - yes Open
1778 56.779784950041396 -0.739517 -20.636 2 19 18 0.86 0.20 - yes Open
2511 56.836178833386235 -0.837185 -23.5688 3 16 0 0.00 0.00 - yes Open
1776 56.85110481560109 -0.694955 -18.2006 0 19 16 0.76 0.00 - yes Open
1771 57.31615126997281 -0.932011 -24.247 2 18 16 0.76 0.20 - yes Current
2506 57.52170037018265 -0.793715 -22.691 3 15 0 0.00 0.00 - yes Open
1863 57.59809028730185 -0.89876 -26.375 3 18 0 0.00 0.00 - yes Open
1854 57.75508683658262 -0.974356 -27.3918 2 18 0 0.00 0.00 - yes Open
1864 58.08813499175179 -0.767908 -21.731 1 17 0 0.00 0.00 - yes Open
1773 58.49758287988025 -0.763956 -24.47 1 18 17 0.81 0.20 - yes Open
1858 58.8597175338021 -0.981518 -26.8425 3 17 0 0.00 0.00 - yes Open
667 60.42742215940044 -0.63983 -9.58648 2 20 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.247kcal/mol
Ligand efficiency (LE) -0.8082kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.796
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 30HA

Physicochemical properties

Molecular weight 398.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.81
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 22.38kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 95.86kcal/mol
Minimised FF energy 73.47kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.