FAIRMol

OSA_Lib_265

Pose ID 1692 Compound 128 Pose 1692

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.650 kcal/mol/HA) ✓ Good fit quality (FQ -6.55) ✗ Very high strain energy (24.5 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-22.735
kcal/mol
LE
-0.650
kcal/mol/HA
Fit Quality
-6.55
FQ (Leeson)
HAC
35
heavy atoms
MW
473
Da
LogP
3.71
cLogP
Strain ΔE
24.5 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 24.5 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 2 Clashes 9 Severe clashes 1
Final rank57.129558873322104Score-22.7347
Inter norm-0.704416Intra norm0.0548541
Top1000noExcludedyes
Contacts18H-bonds2
Artifact reasonexcluded; geometry warning; 18 clashes; 1 protein clash
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap17Native recall0.81
Jaccard0.77RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1690 4.139253699145183 -0.640127 -21.8229 0 18 16 0.76 0.00 - no Open
2393 4.556645021606059 -0.574573 -20.3252 0 14 0 0.00 0.00 - no Open
1686 4.765956123115348 -0.701663 -23.238 1 18 16 0.76 0.00 - no Open
2394 5.092747333470552 -0.61752 -20.4453 1 16 0 0.00 0.00 - no Open
2397 5.164233783323646 -0.52205 -18.6943 0 15 0 0.00 0.00 - no Open
2388 5.224683613549873 -0.568704 -21.1131 1 15 0 0.00 0.00 - no Open
2395 5.535991576416797 -0.618868 -20.9122 2 14 0 0.00 0.00 - no Open
1691 5.6528616715540165 -0.625081 -20.2919 0 18 16 0.76 0.00 - no Open
1689 5.793471843964305 -0.550151 -17.1909 0 17 15 0.71 0.00 - no Open
1685 6.007538655271793 -0.628033 -24.0747 0 18 15 0.71 0.00 - no Open
2389 6.207081991294748 -0.561869 -20.5457 1 14 0 0.00 0.00 - no Open
2390 6.6761583065321135 -0.6451 -21.2028 1 16 0 0.00 0.00 - no Open
1687 9.103784615043438 -0.564845 -19.7451 0 18 15 0.71 0.00 - no Open
2392 54.817570671989 -0.615461 -20.7388 1 15 0 0.00 0.00 - no Open
2398 5.941656091052088 -0.555668 -18.5058 0 16 0 0.00 0.00 - yes Open
2396 8.048595874523157 -0.68237 -22.9115 2 17 0 0.00 0.00 - yes Open
1688 55.92799797916076 -0.687967 -22.2792 2 18 17 0.81 0.00 - yes Open
1692 57.129558873322104 -0.704416 -22.7347 2 18 17 0.81 0.00 - yes Current
2391 57.13284752357958 -0.647544 -21.1325 2 13 0 0.00 0.00 - yes Open
2399 58.20936197376648 -0.612942 -20.666 2 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.735kcal/mol
Ligand efficiency (LE) -0.6496kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.552
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 35HA

Physicochemical properties

Molecular weight 472.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.71
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 24.52kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 113.17kcal/mol
Minimised FF energy 88.65kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.