FAIRMol

OSA_Lib_253

Pose ID 1664 Compound 164 Pose 1664

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.606 kcal/mol/HA) ✓ Good fit quality (FQ -6.11) ✗ Very high strain energy (62.2 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-21.211
kcal/mol
LE
-0.606
kcal/mol/HA
Fit Quality
-6.11
FQ (Leeson)
HAC
35
heavy atoms
MW
475
Da
LogP
1.53
cLogP
Strain ΔE
62.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 62.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 6 Severe clashes 1
Final rank7.8779855370982705Score-21.2107
Inter norm-0.67146Intra norm0.0654404
Top1000noExcludedyes
Contacts17H-bonds1
Artifact reasonexcluded; geometry warning; 12 clashes; 1 protein clash; high strain Δ 56.4
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap17Native recall0.81
Jaccard0.81RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1662 4.350384725323136 -0.738174 -24.6084 1 17 17 0.81 0.00 - no Open
1667 4.844045954796032 -0.700366 -19.294 1 19 17 0.81 0.00 - no Open
1668 4.859384716406591 -0.640292 -21.3225 1 16 13 0.62 0.20 - no Open
1671 5.605918802242034 -0.60581 -20.7046 1 20 17 0.81 0.20 - no Open
1661 7.763985129702788 -0.608674 -17.1888 1 21 18 0.86 0.00 - no Open
1670 54.960284209602236 -0.604768 -18.8776 1 17 16 0.76 0.00 - no Open
1664 7.8779855370982705 -0.67146 -21.2107 1 17 17 0.81 0.00 - yes Current
1672 54.55062236852084 -0.585962 -19.8579 1 17 17 0.81 0.00 - yes Open
1669 55.71954481361269 -0.595588 -21.8651 1 17 17 0.81 0.00 - yes Open
1666 56.025489933285584 -0.713076 -18.0676 1 21 18 0.86 0.00 - yes Open
1665 57.1778127653425 -0.559432 -16.0845 2 21 18 0.86 0.00 - yes Open
1663 58.99218056414671 -0.623854 -20.1822 1 22 19 0.90 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.211kcal/mol
Ligand efficiency (LE) -0.6060kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.113
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 35HA

Physicochemical properties

Molecular weight 474.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.53
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 62.18kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 264.28kcal/mol
Minimised FF energy 202.10kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.