FAIRMol

OSA_Lib_272

Pose ID 15893 Compound 1842 Pose 696

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.747 kcal/mol/HA) ✓ Good fit quality (FQ -7.34) ✗ Very high strain energy (24.4 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-23.888
kcal/mol
LE
-0.747
kcal/mol/HA
Fit Quality
-7.34
FQ (Leeson)
HAC
32
heavy atoms
MW
435
Da
LogP
0.65
cLogP
Strain ΔE
24.4 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 2 Severe clashes 0
Final rank3.610981735712587Score-23.8878
Inter norm-0.758568Intra norm0.0120745
Top1000noExcludedno
Contacts16H-bonds1
Artifact reasongeometry warning; 13 clashes; 2 protein contact clashes; high strain Δ 26.9
ResiduesA:NDP301;B:ARG48;B:ASP52;B:ILE45;B:LEU94;B:MET53;B:PHE56;B:PHE91;B:PRO88;B:SER44;B:SER86;B:THR83;B:TRP47;B:VAL156;B:VAL49;B:VAL87

Protein summary

511 residues
Protein targetT09Atoms8170
Residues511Chains2
Residue summaryLEU:1064; ARG:840; LYS:572; GLU:570; VAL:528; PHE:460; ILE:456; ALA:440; PRO:420; THR:406; TYR:357; ASP:312; GLN:289; ASN:238; SER:231; GLY:224

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts21
PoseOpen native poseH-bonds9
IFP residuesA:NDP301; B:ALA32; B:ARG97; B:ASP52; B:GLY157; B:ILE45; B:LEU94; B:LYS57; B:MET53; B:PHE55; B:PHE56; B:PHE91; B:PRO88; B:SER86; B:THR180; B:THR83; B:TYR162; B:VAL156; B:VAL30; B:VAL31; B:VAL87
Current overlap12Native recall0.57
Jaccard0.48RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
696 3.610981735712587 -0.758568 -23.8878 1 16 12 0.57 0.00 - no Current
693 4.085602005855498 -0.704945 -23.1113 1 20 17 0.81 0.00 - no Open
697 4.163423230648344 -0.854036 -24.2387 1 20 18 0.86 0.00 - no Open
685 4.23461607874702 -0.832023 -24.9795 1 21 18 0.86 0.00 - no Open
686 4.347906685773361 -0.554062 -15.8077 1 11 8 0.38 0.00 - no Open
688 4.602213466082693 -0.646611 -14.8482 1 18 14 0.67 0.00 - no Open
694 5.267078630146593 -0.793475 -24.3561 1 19 18 0.86 0.00 - no Open
687 53.77478225739354 -0.736545 -23.5602 1 17 16 0.76 0.00 - no Open
689 54.11364938603942 -0.708001 -20.9342 1 15 13 0.62 0.00 - no Open
690 54.125530115725724 -0.921161 -28.0447 1 20 18 0.86 0.00 - no Open
691 54.143308804176705 -0.520913 -15.2246 1 10 7 0.33 0.17 - no Open
692 54.712771389708934 -0.537902 -17.0126 1 13 9 0.43 0.00 - no Open
699 5.002453438480102 -0.774088 -20.9243 2 17 17 0.81 0.00 - yes Open
700 5.572610449209327 -0.622267 -19.1936 1 18 14 0.67 0.00 - yes Open
698 55.32201350023294 -0.564031 -16.8084 0 12 6 0.29 0.00 - yes Open
695 56.64804480159266 -0.599192 -19.9787 1 11 8 0.38 0.17 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.888kcal/mol
Ligand efficiency (LE) -0.7465kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.341
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 434.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.65
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 24.45kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 235.18kcal/mol
Minimised FF energy 210.73kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.