FAIRMol

OSA_Lib_227

Pose ID 1484 Compound 172 Pose 1484

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.475 kcal/mol/HA) ✓ Good fit quality (FQ -4.83) ✗ Very high strain energy (27.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-17.097
kcal/mol
LE
-0.475
kcal/mol/HA
Fit Quality
-4.83
FQ (Leeson)
HAC
36
heavy atoms
MW
489
Da
LogP
2.06
cLogP
Strain ΔE
27.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 27.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 13 Severe clashes 3
Final rank59.82543377216085Score-17.0973
Inter norm-0.521391Intra norm0.0464658
Top1000noExcludedyes
Contacts17H-bonds1
Artifact reasonexcluded; geometry warning; 13 clashes; 3 protein clashes
ResiduesA:ALA10;A:ASP22;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:THR137;A:THR57;A:TYR34;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap14Native recall0.67
Jaccard0.58RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1493 4.436227231282095 -0.69089 -25.5895 1 20 17 0.81 0.00 - no Open
1477 4.6014129751987625 -0.660838 -22.7681 0 20 17 0.81 0.00 - no Open
1495 4.662853712023105 -0.606409 -23.1152 1 20 17 0.81 0.00 - no Open
1487 4.885390810668738 -0.615988 -21.32 0 20 17 0.81 0.00 - no Open
1470 5.125298776994811 -0.639317 -21.7068 1 19 16 0.76 0.00 - no Open
1480 5.2195099021393245 -0.58901 -20.786 0 17 15 0.71 0.00 - no Open
1482 5.229026063789104 -0.609474 -19.0643 0 16 13 0.62 0.00 - no Open
1489 5.744689911396554 -0.648348 -22.5503 1 17 15 0.71 0.20 - no Open
1490 5.792566717545938 -0.600301 -23.0593 0 16 13 0.62 0.00 - no Open
1472 5.81085638361404 -0.687729 -23.5496 1 18 17 0.81 0.20 - no Open
1496 6.032172607963344 -0.534558 -19.6404 0 20 17 0.81 0.00 - no Open
1481 6.972896016620622 -0.710599 -21.7006 1 19 16 0.76 0.00 - no Open
1486 55.06858250933098 -0.594794 -17.609 1 19 16 0.76 0.00 - no Open
1478 6.247720023293538 -0.707476 -20.7339 1 18 16 0.76 0.00 - yes Open
1469 6.664881426753806 -0.5965 -19.7656 0 21 18 0.86 0.00 - yes Open
1483 9.729741189547976 -0.557839 -17.1565 1 17 17 0.81 0.20 - yes Open
1479 55.381965180018014 -0.663129 -23.4074 1 17 15 0.71 0.20 - yes Open
1494 55.49501787708691 -0.639752 -18.2612 0 17 13 0.62 0.00 - yes Open
1485 56.22822988942302 -0.641435 -19.3369 1 19 18 0.86 0.00 - yes Open
1474 56.58695063875411 -0.691658 -24.7988 1 18 18 0.86 0.00 - yes Open
1488 56.75211749384185 -0.620956 -24.7199 1 17 17 0.81 0.00 - yes Open
1473 57.317364973581775 -0.574226 -18.2593 1 18 17 0.81 0.20 - yes Open
1471 57.48824315941614 -0.678132 -24.7077 1 17 17 0.81 0.00 - yes Open
1492 57.89452978962589 -0.772931 -19.0049 1 20 16 0.76 0.00 - yes Open
1475 57.91227650358714 -0.638687 -20.0354 3 20 17 0.81 0.20 - yes Open
1491 59.73448931696643 -0.655337 -14.4505 1 20 17 0.81 0.00 - yes Open
1484 59.82543377216085 -0.521391 -17.0973 1 17 14 0.67 0.20 - yes Current
1476 60.553477368626375 -0.599194 -19.4365 3 20 17 0.81 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -17.097kcal/mol
Ligand efficiency (LE) -0.4749kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.827
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 36HA

Physicochemical properties

Molecular weight 488.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.06
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 27.10kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 198.67kcal/mol
Minimised FF energy 171.57kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.