FAIRMol

OSA_Lib_222

Pose ID 1432 Compound 183 Pose 1432

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good LE (-0.320 kcal/mol/HA) ✓ Good fit quality (FQ -3.22) ✗ Very high strain energy (38.5 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-11.188
kcal/mol
LE
-0.320
kcal/mol/HA
Fit Quality
-3.22
FQ (Leeson)
HAC
35
heavy atoms
MW
478
Da
LogP
1.38
cLogP
Strain ΔE
38.5 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: good
Geometry reliability: low
Reason: geometry warning, clashes, strain 38.5 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 0 Clashes 8 Severe clashes 1
Final rank8.044199703719837Score-11.1879
Inter norm-0.56172Intra norm0.242065
Top1000noExcludedyes
Contacts17H-bonds2
Artifact reasonexcluded; geometry warning; 16 clashes; 1 protein clash; high strain Δ 32.6
ResiduesA:ALA10;A:ARG29;A:ASN65;A:ASP22;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO26;A:PRO27;A:PRO62;A:TRP25

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap12Native recall0.57
Jaccard0.46RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1421 4.507450501626563 -0.597193 -16.8932 0 18 15 0.71 0.00 - no Open
1426 5.704592347039669 -0.572579 -8.02978 1 18 15 0.71 0.00 - no Open
1433 6.140176582882947 -0.636588 -20.8592 1 19 17 0.81 0.00 - no Open
1434 6.236590408376431 -0.515547 -10.8775 2 19 15 0.71 0.20 - no Open
1422 6.293581608737499 -0.528888 -18.2267 0 20 16 0.76 0.00 - no Open
1425 55.424855903405 -0.558437 -17.3614 1 19 15 0.71 0.00 - no Open
1428 55.47899451594846 -0.727061 -15.9633 2 18 14 0.67 0.00 - no Open
1424 56.78165473858708 -0.532831 -16.8104 0 21 17 0.81 0.00 - no Open
1432 8.044199703719837 -0.56172 -11.1879 2 17 12 0.57 0.20 - yes Current
1436 56.96879084411105 -0.766017 -16.0094 2 18 14 0.67 0.00 - yes Open
1431 57.34162299909664 -0.613912 -19.4608 1 16 14 0.67 0.20 - yes Open
1430 57.42239171600288 -0.59804 -20.3206 1 17 14 0.67 0.00 - yes Open
1427 57.45506349585565 -0.640829 -22.6474 1 19 16 0.76 0.00 - yes Open
1435 57.59561729741003 -0.566975 -17.8114 2 12 9 0.43 0.20 - yes Open
1429 57.91177452793163 -0.499876 -16.4034 0 19 15 0.71 0.00 - yes Open
1423 58.272609059514394 -0.587379 -17.6569 0 22 20 0.95 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -11.188kcal/mol
Ligand efficiency (LE) -0.3197kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -3.224
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 35HA

Physicochemical properties

Molecular weight 477.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.38
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 38.54kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 174.84kcal/mol
Minimised FF energy 136.29kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.