FAIRMol

MK65

Pose ID 13662 Compound 1328 Pose 809

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.286 kcal/mol/HA) ✓ Good fit quality (FQ -11.17) ✓ Strong H-bond network (8 bonds) ✗ High strain energy (19.4 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-28.294
kcal/mol
LE
-1.286
kcal/mol/HA
Fit Quality
-11.17
FQ (Leeson)
HAC
22
heavy atoms
MW
338
Da
LogP
4.01
cLogP
Strain ΔE
19.4 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 8 Hydrophobic 21 π–π 2 Clashes 8 Severe clashes 0
Final rank2.862657882285701Score-28.2945
Inter norm-1.46501Intra norm0.178893
Top1000noExcludedno
Contacts13H-bonds8
Artifact reasongeometry warning; 3 clashes; 8 protein contact clashes; high strain Δ 27.3
ResiduesA:ARG14;A:ASP161;A:CYS168;A:GLY205;A:LEU208;A:LEU209;A:MET213;A:NAP301;A:PHE97;A:PRO210;A:TRP221;A:TYR174;A:VAL206

Protein summary

258 residues
Protein targetT08Atoms3881
Residues258Chains2
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap13Native recall0.68
Jaccard0.68RMSD-
H-bond strict1Strict recall0.17
H-bond same residue+role1Role recall0.20
H-bond same residue3Residue recall0.60

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
709 2.428301583564728 -1.28615 -25.8079 8 17 16 0.84 0.60 - no Open
809 2.862657882285701 -1.46501 -28.2945 8 13 13 0.68 0.20 - no Current
1047 2.8875597911216913 -0.92973 -17.5668 5 12 0 0.00 0.00 - no Open
984 3.209858072408278 -1.09517 -21.6566 7 17 0 0.00 0.00 - no Open
810 3.223976694411096 -1.3611 -23.4229 10 13 13 0.68 0.20 - no Open
808 4.091499979284675 -1.48592 -26.126 8 13 13 0.68 0.20 - no Open
712 2.9662881653437343 -1.35137 -27.1477 6 14 14 0.74 0.40 - yes Open
711 3.4722246272024035 -1.15195 -20.6805 7 12 12 0.63 0.40 - yes Open
1045 4.248139559050531 -1.21411 -23.6042 6 14 0 0.00 0.00 - yes Open
985 5.054451581641908 -0.997149 -19.777 6 16 0 0.00 0.00 - yes Open
1048 5.217677319409357 -1.0922 -21.3075 6 16 0 0.00 0.00 - yes Open
710 5.349640619638379 -1.28432 -21.1214 8 12 12 0.63 0.40 - yes Open
982 6.247471639250551 -1.05281 -18.9823 7 17 0 0.00 0.00 - yes Open
983 6.3984681808428725 -1.00281 -18.1211 7 17 0 0.00 0.00 - yes Open
807 7.197939495020938 -1.28687 -26.03 5 16 15 0.79 0.40 - yes Open
1046 7.862624388908564 -1.22425 -24.6194 6 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -28.294kcal/mol
Ligand efficiency (LE) -1.2861kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -11.166
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 22HA

Physicochemical properties

Molecular weight 338.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.01
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 19.38kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 41.33kcal/mol
Minimised FF energy 21.95kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.