FAIRMol

OSA_Lib_202

Pose ID 1364 Compound 273 Pose 1364

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.561 kcal/mol/HA) ✓ Good fit quality (FQ -5.66) ✗ Very high strain energy (25.3 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-19.647
kcal/mol
LE
-0.561
kcal/mol/HA
Fit Quality
-5.66
FQ (Leeson)
HAC
35
heavy atoms
MW
471
Da
LogP
4.21
cLogP
Strain ΔE
25.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 25.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 15 Severe clashes 1
Final rank58.691692518465146Score-19.647
Inter norm-0.637471Intra norm0.0761284
Top1000noExcludedyes
Contacts18H-bonds1
Artifact reasonexcluded; geometry warning; 16 clashes; 1 protein clash
ResiduesA:ALA10;A:ASP22;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:SER60;A:THR137;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap16Native recall0.76
Jaccard0.70RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1361 5.285932816292426 -0.583383 -19.2555 3 17 14 0.67 0.20 - no Open
1359 5.645237162559839 -0.54001 -18.3822 0 18 18 0.86 0.00 - no Open
516 5.9317471941878885 -0.639332 -18.9075 6 15 0 0.00 0.00 - no Open
519 6.030492630509353 -0.618127 -12.4709 7 13 0 0.00 0.00 - no Open
1357 6.033288432484866 -0.618468 -21.7834 3 14 11 0.52 0.20 - no Open
517 6.9143397434043985 -0.686772 -20.3283 7 14 0 0.00 0.00 - no Open
515 57.76441284196875 -0.73519 -17.1413 7 14 0 0.00 0.00 - no Open
512 56.27641658683974 -0.644971 -17.2738 8 13 0 0.00 0.00 - yes Open
514 58.02966704469649 -0.706296 -21.0217 7 15 0 0.00 0.00 - yes Open
1360 58.20375068390502 -0.518137 -11.1156 2 21 19 0.90 0.00 - yes Open
1358 58.22189820618301 -0.680031 -15.9048 2 19 17 0.81 0.00 - yes Open
513 58.56527856047408 -0.726922 -23.7588 6 15 0 0.00 0.00 - yes Open
1364 58.691692518465146 -0.637471 -19.647 1 18 16 0.76 0.00 - yes Current
1363 58.73527100549721 -0.685777 -18.2544 2 23 19 0.90 0.00 - yes Open
518 58.81415690039258 -0.709034 -21.9524 7 13 0 0.00 0.00 - yes Open
1362 60.668165393281505 -0.729934 -11.1864 2 21 19 0.90 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -19.647kcal/mol
Ligand efficiency (LE) -0.5613kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.662
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 35HA

Physicochemical properties

Molecular weight 470.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.21
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 25.30kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 83.55kcal/mol
Minimised FF energy 58.24kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.