FAIRMol

KB_chagas_47

Pose ID 13426 Compound 824 Pose 573

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.787 kcal/mol/HA) ✓ Good fit quality (FQ -6.95) ✗ Very high strain energy (25.2 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-18.107
kcal/mol
LE
-0.787
kcal/mol/HA
Fit Quality
-6.95
FQ (Leeson)
HAC
23
heavy atoms
MW
352
Da
LogP
3.58
cLogP
Strain ΔE
25.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 25.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 6 Severe clashes 1
Final rank4.96742283390219Score-18.1066
Inter norm-1.0902Intra norm0.302954
Top1000noExcludedyes
Contacts16H-bonds1
Artifact reasonexcluded; geometry warning; 9 clashes; 1 protein clash; high strain Δ 25.7
ResiduesA:ARG14;A:ASP161;A:CYS168;A:GLY205;A:LEU208;A:LEU209;A:LEU263;A:MET163;A:NAP301;A:PHE97;A:PRO210;A:SER207;A:SER95;A:TRP221;A:TYR174;A:VAL206

Protein summary

258 residues
Protein targetT08Atoms3881
Residues258Chains2
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap14Native recall0.74
Jaccard0.67RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
232 2.834794242434497 -1.02933 -17.7647 0 11 0 0.00 0.00 - no Open
235 3.1016599288773388 -0.942173 -17.8202 0 13 0 0.00 0.00 - no Open
574 3.3728629943587816 -1.36419 -26.244 2 15 14 0.74 0.20 - no Open
572 3.8503173755325215 -1.11654 -19.9403 3 10 8 0.42 0.40 - no Open
233 3.9172101203965464 -1.02313 -17.9656 0 13 0 0.00 0.00 - no Open
230 4.521749855716406 -0.912026 -16.9128 0 12 0 0.00 0.00 - no Open
234 4.557625005324844 -0.962951 -16.7474 0 12 0 0.00 0.00 - yes Open
573 4.96742283390219 -1.0902 -18.1066 1 16 14 0.74 0.00 - yes Current
231 55.328014273835905 -0.934761 -16.9919 0 11 0 0.00 0.00 - yes Open
575 56.143906454773145 -1.22344 -24.7009 2 15 13 0.68 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -18.107kcal/mol
Ligand efficiency (LE) -0.7872kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.948
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 23HA

Physicochemical properties

Molecular weight 352.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.58
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 25.17kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 61.68kcal/mol
Minimised FF energy 36.52kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.