FAIRMol

OHD_TB2021_31

Pose ID 13053 Compound 1600 Pose 200

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Promising Reasonable quality metrics. Warrants further investigation.
✓ Excellent LE (-1.264 kcal/mol/HA) ✓ Good fit quality (FQ -11.64) ✓ Strong H-bond network (9 bonds) ✗ Moderate strain (8.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-32.851
kcal/mol
LE
-1.264
kcal/mol/HA
Fit Quality
-11.64
FQ (Leeson)
HAC
26
heavy atoms
MW
344
Da
LogP
2.51
cLogP
Strain ΔE
8.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes

Interaction summary

Collapsible panels
H-bonds 9 Hydrophobic 24 π–π 4 Clashes 16 Severe clashes 1
Final rank7.192673937326427Score-32.8511
Inter norm-1.22639Intra norm-0.0371144
Top1000noExcludedyes
Contacts19H-bonds9
Artifact reasonexcluded; geometry warning; 11 clashes; 1 protein clash
ResiduesA:ALA96;A:ARG14;A:ASN127;A:ASP161;A:CYS168;A:GLY205;A:LEU208;A:LEU209;A:LEU263;A:LYS178;A:MET163;A:MET213;A:NAP301;A:PHE97;A:PRO210;A:SER95;A:TRP221;A:TYR174;A:VAL206

Protein summary

258 residues
Protein targetT08Atoms3881
Residues258Chains2
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap15Native recall0.79
Jaccard0.65RMSD-
H-bond strict3Strict recall0.50
H-bond same residue+role2Role recall0.40
H-bond same residue2Residue recall0.40

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
193 2.341573079589889 -0.795871 -19.8565 3 10 0 0.00 0.00 - no Open
187 2.600580136268462 -1.00176 -23.1171 3 17 0 0.00 0.00 - no Open
192 2.612595909471465 -0.814557 -22.3807 3 10 0 0.00 0.00 - no Open
186 3.181781192158638 -1.01831 -25.6436 2 16 0 0.00 0.00 - no Open
188 3.1859197969722253 -0.998321 -23.6116 3 16 0 0.00 0.00 - no Open
128 3.566475201443353 -1.2388 -31.1169 4 21 0 0.00 0.00 - no Open
201 3.679863303157364 -1.32526 -34.0392 8 17 13 0.68 0.60 - no Open
194 3.742749019480482 -0.789796 -19.532 3 10 0 0.00 0.00 - no Open
242 3.881589315785158 -0.722011 -20.936 5 12 0 0.00 0.00 - no Open
202 5.603465179791285 -1.38948 -29.4696 7 16 11 0.58 0.60 - yes Open
200 7.192673937326427 -1.22639 -32.8511 9 19 15 0.79 0.40 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -32.851kcal/mol
Ligand efficiency (LE) -1.2635kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -11.641
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 344.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.51
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 8.43kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 75.80kcal/mol
Minimised FF energy 67.37kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.