FAIRMol

Z49894143

Pose ID 12801 Compound 1352 Pose 2363

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.365 kcal/mol/HA) ✓ Good fit quality (FQ -12.04) ✗ High strain energy (19.1 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-31.389
kcal/mol
LE
-1.365
kcal/mol/HA
Fit Quality
-12.04
FQ (Leeson)
HAC
23
heavy atoms
MW
343
Da
LogP
4.67
cLogP
Strain ΔE
19.1 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 7 Severe clashes 0
Final rank3.6021220444997133Score-31.3889
Inter norm-1.28928Intra norm-0.0754483
Top1000noExcludedno
Contacts13H-bonds1
Artifact reasongeometry warning; 9 clashes; 7 protein contact clashes; high strain Δ 22.9
ResiduesA:ARG14;A:ASP161;A:CYS168;A:GLY205;A:LEU208;A:LEU209;A:MET213;A:NAP301;A:PHE97;A:PRO210;A:TRP221;A:TYR174;A:VAL206

Protein summary

275 residues
Protein targetT07Atoms3932
Residues275Chains3
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap13Native recall0.68
Jaccard0.68RMSD-
H-bond strict1Strict recall0.17
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2362 2.9650887442105436 -1.13891 -30.3459 1 12 12 0.63 0.00 - no Open
2360 3.0206159107306734 -1.13801 -25.1298 1 12 12 0.63 0.00 - no Open
2363 3.6021220444997133 -1.28928 -31.3889 1 13 13 0.68 0.20 - no Current
2361 3.6221867520846573 -1.13393 -25.0201 1 13 13 0.68 0.20 - no Open
3019 4.565328450590989 -0.947343 -24.4468 6 11 0 0.00 0.00 - no Open
3018 6.265726631676909 -1.08382 -25.5871 7 15 0 0.00 0.00 - yes Open
3017 6.527330848851234 -0.840207 -19.3993 3 15 0 0.00 0.00 - yes Open
3020 8.411018072258297 -0.86015 -22.7911 5 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -31.389kcal/mol
Ligand efficiency (LE) -1.3647kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -12.045
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 23HA

Physicochemical properties

Molecular weight 342.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.67
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 19.11kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 50.80kcal/mol
Minimised FF energy 31.69kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.