FAIRMol

Z49539235

Pose ID 12556 Compound 1290 Pose 2118

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.614 kcal/mol/HA) ✓ Good fit quality (FQ -5.03) ✗ Very high strain energy (27.3 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-11.666
kcal/mol
LE
-0.614
kcal/mol/HA
Fit Quality
-5.03
FQ (Leeson)
HAC
19
heavy atoms
MW
321
Da
LogP
2.43
cLogP
Strain ΔE
27.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 27.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 20 π–π 2 Clashes 8 Severe clashes 1
Final rank5.976793057249998Score-11.6663
Inter norm-1.0197Intra norm0.405686
Top1000noExcludedyes
Contacts13H-bonds1
Artifact reasonexcluded; geometry warning; 9 clashes; 1 protein clash; high strain Δ 32.7
ResiduesA:ARG14;A:GLY205;A:LEU208;A:LEU209;A:LEU263;A:MET163;A:NAP301;A:PHE97;A:PRO210;A:SER95;A:TRP221;A:TYR174;A:VAL206

Protein summary

275 residues
Protein targetT07Atoms3932
Residues275Chains3
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap11Native recall0.58
Jaccard0.52RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2117 1.3448581504504311 -1.33434 -26.5502 6 13 13 0.68 0.20 - no Open
2115 1.4273602231327094 -1.57092 -30.5567 6 13 13 0.68 0.40 - no Open
2119 1.7902050583631977 -1.39142 -27.7622 4 13 13 0.68 0.20 - no Open
2111 2.059366333586598 -1.6235 -31.4971 6 15 14 0.74 0.40 - no Open
2114 2.78249284218905 -1.0947 -22.3777 3 17 14 0.74 0.40 - no Open
2113 2.8591259614089726 -1.6099 -31.5095 5 13 13 0.68 0.40 - no Open
2116 3.3561098991350917 -1.19755 -19.7952 1 14 12 0.63 0.20 - yes Open
2112 4.811622542538363 -1.09673 -21.0691 3 15 12 0.63 0.20 - yes Open
2118 5.976793057249998 -1.0197 -11.6663 1 13 11 0.58 0.20 - yes Current
2110 6.024028625348568 -1.29141 -24.3603 6 14 12 0.63 0.60 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -11.666kcal/mol
Ligand efficiency (LE) -0.6140kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.033
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 19HA

Physicochemical properties

Molecular weight 321.2Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.43
Lipinski: ≤ 5
Rotatable bonds 2

Conformational strain (MMFF94s)

Strain energy (ΔE) 27.31kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 61.34kcal/mol
Minimised FF energy 34.03kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.