FAIRMol

OSA_Lib_133

Pose ID 1250 Compound 225 Pose 1250

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.699 kcal/mol/HA) ✓ Good fit quality (FQ -6.93) ✗ Very high strain energy (33.6 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-23.051
kcal/mol
LE
-0.699
kcal/mol/HA
Fit Quality
-6.93
FQ (Leeson)
HAC
33
heavy atoms
MW
448
Da
LogP
1.80
cLogP
Strain ΔE
33.6 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 33.6 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 4 Severe clashes 1
Final rank55.25138654316312Score-23.0511
Inter norm-0.706578Intra norm0.00805847
Top1000noExcludedyes
Contacts21H-bonds1
Artifact reasonexcluded; geometry warning; 15 clashes; 1 protein clash
ResiduesA:ALA10;A:ARG29;A:ASN65;A:ASP22;A:GLN36;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.75RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1016 3.6903788952797765 -0.476658 -19.7047 4 12 0 0.00 0.00 - no Open
1015 4.336715025239418 -0.476824 -16.4556 3 13 0 0.00 0.00 - no Open
1011 4.677775971132904 -0.490975 -16.5462 3 14 0 0.00 0.00 - no Open
1256 4.87390419593541 -0.598743 -22.6002 0 16 14 0.67 0.00 - no Open
1253 5.744303461001272 -0.541821 -17.0864 1 14 11 0.52 0.20 - no Open
1254 6.657045936166917 -0.566659 -19.5657 0 20 18 0.86 0.00 - no Open
1014 53.77516763994396 -0.401003 -11.6208 1 12 0 0.00 0.00 - no Open
1010 54.36786590845734 -0.563195 -19.5894 3 10 0 0.00 0.00 - no Open
1255 55.20943744404354 -0.742831 -26.5815 1 23 19 0.90 0.00 - no Open
1009 55.269055794228294 -0.396214 -15.0353 0 10 0 0.00 0.00 - no Open
1249 55.903832911816465 -0.576255 -23.5896 0 17 16 0.76 0.00 - no Open
1250 55.25138654316312 -0.706578 -23.0511 1 21 18 0.86 0.00 - yes Current
1012 55.27958761014378 -0.534138 -15.972 2 12 0 0.00 0.00 - yes Open
1251 57.356232960664 -0.658721 -19.8679 1 19 16 0.76 0.00 - yes Open
1013 58.320955243854094 -0.441868 -11.1203 2 13 0 0.00 0.00 - yes Open
1252 59.843782502125954 -0.546685 -8.16592 1 20 18 0.86 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.051kcal/mol
Ligand efficiency (LE) -0.6985kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.931
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 33HA

Physicochemical properties

Molecular weight 447.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.80
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 33.63kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 128.87kcal/mol
Minimised FF energy 95.23kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.