FAIRMol

Z275164792

Pose ID 11934 Compound 1348 Pose 1496

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.512 kcal/mol/HA) ✓ Good fit quality (FQ -12.39) ✓ Good H-bonds (3 bonds) ✗ High strain energy (10.3 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-28.724
kcal/mol
LE
-1.512
kcal/mol/HA
Fit Quality
-12.39
FQ (Leeson)
HAC
19
heavy atoms
MW
321
Da
LogP
2.63
cLogP
Strain ΔE
10.3 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 2 Clashes 6 Severe clashes 0
Final rank2.8866079816749814Score-28.7244
Inter norm-1.53112Intra norm0.019307
Top1000noExcludedno
Contacts13H-bonds3
Artifact reasongeometry warning; 11 clashes; 6 protein contact clashes; moderate strain Δ 12.3
ResiduesA:ARG14;A:ASP161;A:CYS168;A:LEU208;A:LEU209;A:MET213;A:NAP301;A:PHE97;A:PRO210;A:SER207;A:TRP221;A:TYR174;A:VAL206

Protein summary

275 residues
Protein targetT07Atoms3932
Residues275Chains3
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap13Native recall0.68
Jaccard0.68RMSD-
H-bond strict1Strict recall0.17
H-bond same residue+role1Role recall0.20
H-bond same residue3Residue recall0.60

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1496 2.8866079816749814 -1.53112 -28.7244 3 13 13 0.68 0.20 - no Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -28.724kcal/mol
Ligand efficiency (LE) -1.5118kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -12.392
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 19HA

Physicochemical properties

Molecular weight 321.2Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.63
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 10.31kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 57.15kcal/mol
Minimised FF energy 46.83kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.