FAIRMol

OHD_Leishmania_407

Pose ID 10555 Compound 474 Pose 117

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.219 kcal/mol/HA) ✓ Good fit quality (FQ -10.93) ✓ Strong H-bond network (6 bonds) ✗ High strain energy (14.3 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-29.266
kcal/mol
LE
-1.219
kcal/mol/HA
Fit Quality
-10.93
FQ (Leeson)
HAC
24
heavy atoms
MW
365
Da
LogP
2.51
cLogP
Strain ΔE
14.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 14.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 6 Hydrophobic 24 π–π 4 Clashes 6 Severe clashes 0
Final rank3.3037872853401975Score-29.2661
Inter norm-1.18971Intra norm-0.0297105
Top1000noExcludedno
Contacts14H-bonds6
Artifact reasongeometry warning; 12 clashes; 6 protein contact clashes; moderate strain Δ 13.5
ResiduesA:ARG14;A:ASP161;A:CYS168;A:LEU208;A:LEU209;A:MET213;A:NAP301;A:PHE171;A:PHE97;A:PRO210;A:SER95;A:TRP221;A:TYR174;A:VAL206

Protein summary

275 residues
Protein targetT07Atoms3932
Residues275Chains3
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap14Native recall0.74
Jaccard0.74RMSD-
H-bond strict3Strict recall0.50
H-bond same residue+role2Role recall0.40
H-bond same residue2Residue recall0.40

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
172 2.9583132347911665 -1.20346 -25.7588 10 17 0 0.00 0.00 - no Open
119 3.0411416082296214 -1.18879 -29.0207 6 14 14 0.74 0.40 - no Open
117 3.3037872853401975 -1.18971 -29.2661 6 14 14 0.74 0.40 - no Current
170 4.451495078205778 -1.16923 -25.0891 6 16 0 0.00 0.00 - no Open
118 5.18116131436111 -1.15484 -25.0514 7 12 12 0.63 0.40 - no Open
122 5.471817934988997 -0.743153 -15.0498 5 19 0 0.00 0.00 - no Open
120 5.6539743183894 -1.12904 -24.6433 7 12 12 0.63 0.40 - no Open
171 4.618794082020386 -1.18707 -21.4229 11 16 0 0.00 0.00 - yes Open
173 54.02556249294625 -1.20338 -22.2631 9 16 0 0.00 0.00 - yes Open
123 59.382537021470505 -0.878394 -19.1316 6 19 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -29.266kcal/mol
Ligand efficiency (LE) -1.2194kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -10.928
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 24HA

Physicochemical properties

Molecular weight 365.2Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.51
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 14.31kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy -135.83kcal/mol
Minimised FF energy -150.14kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.