FAIRMol

OHD_Leishmania_135

Pose ID 10526 Compound 645 Pose 88

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-1.132 kcal/mol/HA) ✓ Good fit quality (FQ -11.42) ✓ Strong H-bond network (6 bonds) ✗ Very high strain energy (32.3 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-39.634
kcal/mol
LE
-1.132
kcal/mol/HA
Fit Quality
-11.42
FQ (Leeson)
HAC
35
heavy atoms
MW
480
Da
LogP
1.45
cLogP
Strain ΔE
32.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 32.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 6 Hydrophobic 24 π–π 3 Clashes 4 Severe clashes 1
Final rank6.701023002482439Score-39.6339
Inter norm-1.03729Intra norm-0.0951049
Top1000noExcludedyes
Contacts21H-bonds6
Artifact reasonexcluded; geometry warning; 15 clashes; 1 protein clash; high strain Δ 45.4
ResiduesA:ALA96;A:ARG14;A:ASP161;A:CYS168;A:GLU217;A:GLY205;A:LEU208;A:LEU209;A:LYS178;A:LYS220;A:MET169;A:MET213;A:NAP301;A:PHE171;A:PHE97;A:PRO210;A:SER207;A:SER95;A:TRP221;A:TYR174;A:VAL206

Protein summary

275 residues
Protein targetT07Atoms3932
Residues275Chains3
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap17Native recall0.89
Jaccard0.74RMSD-
H-bond strict5Strict recall0.83
H-bond same residue+role4Role recall0.80
H-bond same residue4Residue recall0.80

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
87 4.643498246436422 -1.05255 -36.6414 7 20 17 0.89 0.80 - no Open
70 5.476196025311045 -0.739124 -24.709 12 22 0 0.00 0.00 - no Open
33 6.480727755154504 -0.81612 -23.4258 7 15 0 0.00 0.00 - no Open
95 7.87152207715595 -0.794446 -29.5766 6 22 0 0.00 0.00 - no Open
88 6.701023002482439 -1.03729 -39.6339 6 21 17 0.89 0.80 - yes Current
86 6.891187406146223 -1.04094 -29.6961 6 20 16 0.84 0.80 - yes Open
69 7.772060174584413 -0.71998 -20.8914 10 21 0 0.00 0.00 - yes Open
71 9.113995759443968 -0.727321 -29.2617 10 22 0 0.00 0.00 - yes Open
32 10.755888868764302 -0.9847 -29.0807 7 16 0 0.00 0.00 - yes Open
94 12.364613215489982 -0.722233 -24.7408 9 21 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -39.634kcal/mol
Ligand efficiency (LE) -1.1324kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -11.422
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 35HA

Physicochemical properties

Molecular weight 479.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.45
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 32.33kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 94.52kcal/mol
Minimised FF energy 62.20kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.