FAIRMol

OHD_Leishmania_125

Pose ID 10495 Compound 1031 Pose 57

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.992 kcal/mol/HA) ✓ Good fit quality (FQ -10.30) ✓ Strong H-bond network (9 bonds) ✗ Very high strain energy (39.2 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-38.703
kcal/mol
LE
-0.992
kcal/mol/HA
Fit Quality
-10.30
FQ (Leeson)
HAC
39
heavy atoms
MW
528
Da
LogP
2.24
cLogP
Strain ΔE
39.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 39.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 9 Hydrophobic 24 π–π 3 Clashes 0 Severe clashes 0
Final rank4.558706331096513Score-38.7032
Inter norm-0.969977Intra norm-0.0224139
Top1000noExcludedno
Contacts19H-bonds9
Artifact reasongeometry warning; 19 clashes; high strain Δ 42.8
ResiduesA:ALA96;A:ARG14;A:ASP161;A:CYS168;A:GLU217;A:LEU208;A:LEU209;A:MET163;A:MET213;A:NAP301;A:PHE171;A:PHE97;A:PRO210;A:PRO99;A:SER207;A:SER95;A:TRP221;A:TYR174;A:VAL206

Protein summary

275 residues
Protein targetT07Atoms3932
Residues275Chains3
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap16Native recall0.84
Jaccard0.73RMSD-
H-bond strict5Strict recall0.83
H-bond same residue+role4Role recall0.80
H-bond same residue4Residue recall0.80

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

No clashes detected for this pose.

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
57 4.558706331096513 -0.969977 -38.7032 9 19 16 0.84 0.80 - no Current
56 5.316952564828583 -0.923397 -38.9963 7 19 16 0.84 0.80 - no Open
58 6.075260472483174 -0.962437 -40.2519 7 19 16 0.84 0.80 - no Open
72 8.918246884165283 -0.598542 -20.7155 12 22 0 0.00 0.00 - no Open
98 9.117215121004701 -0.69453 -22.5704 11 21 0 0.00 0.00 - no Open
8 9.31166288367184 -0.661104 -16.044 3 15 0 0.00 0.00 - no Open
6 11.706246338544839 -0.846386 -25.6976 5 15 0 0.00 0.00 - yes Open
73 14.994885260763583 -0.631646 -24.6039 3 23 0 0.00 0.00 - yes Open
7 15.024825254720277 -0.649781 -20.0045 7 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -38.703kcal/mol
Ligand efficiency (LE) -0.9924kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -10.299
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 39HA

Physicochemical properties

Molecular weight 527.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.24
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 39.15kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 107.19kcal/mol
Minimised FF energy 68.04kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.